Tocris/XD 14/5489/50/50毫克-免疫在线蚂蚁淘旗下平台

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商品详细Tocris/XD 14/5489/50/50毫克

Tocris/XD 14/5489/50/50毫克

商品编号： 5489/50

品牌： Tocris Bioscience

市场价： ¥17580.00

美元价： 10548.00

产地：美国(厂家直采)

公司：

产品分类：多肽

公司分类： peptides

联系Q Q： 3392242852

电话号码： 4000-520-616

电子邮箱： info@ebiomall.com

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商品介绍

Description:BETbromodomaininhibitor

ChemicalName:4-Acetyl-N-[5-[(diethylamino)sulfonyl]-2-hydroxyphenyl]-3-ethyl-5-methyl-1H-pyrrole-2-carboxamide

Purity:≥98%(HPLC)

BIOLOGicalActivityTechnicalDataSolubilityCalculatorsDatasheetsReferences

BiologicalActivity

BETbromodomaininhibitor(K_dvaluesare160,170,380,490,830and850nMforBRD4(1),BRD2(1),BRD3(1),BRD3(2),BRD2(2)andBRD4(2)respectively).AlsoinhibitsBRDT(1),CBP,p300andBRDT(2)(K_dvaluesare1.2,1.6,2.6and3.7μMrespectively).AttenuatesproliferationofHL-60leukemiacellsinvitro.

CompoundLibraries

XD14isalsoofferedaspartoftheTocriscreenPlus.FindoutmoreaboutcompoundlibrariesavailablefromTocris.

TechnicalData

M.Wt	421.51
Formula	C₂₀H₂₇N₃O₅S
Storage	Storeat-20°C
Purity	≥98%(HPLC)
CASNumber	1370888-71-3
PubChemID	52670832
InChIKey	DPBKLIVPNYGQQG-UHFFFAOYSA-N
Smiles	CC1=C(C(C)=O)C(CC)=C(C(NC2=CC(S(N(CC)CC)(=O)=O)=CC=C2O)=O)N1

Thetechnicaldataprovidedaboveisforguidanceonly.ForbatchspecificdatarefertotheCertificateofAnalysis.

AllTocrisproductsareintendedforlaboratoryresearchuseonly.

SolubilityData

	Solvent	MaxConc.mg/mL	MaxConc.mM
Solubility
	DMSO	42.15	100
	ethanol	42.15	100

PreparingStockSolutions

Thefollowingdataisbasedontheproductmolecularweight421.51.Batchspecificmolecularweightsmayvaryfrombatchtobatchduetosolventofhydration,whichwillaffectthesolventvolumesrequiredtopreparestocksolutions.

Concentration/SolventVolume/Mass	1mg	5mg	10mg
1mM	2.37mL	11.86mL	23.72mL
5mM	0.47mL	2.37mL	4.74mL
10mM	0.24mL	1.19mL	2.37mL
50mM	0.05mL	0.24mL	0.47mL

ProductDatasheets

CertificateofAnalysis/ProductDatasheet

SafetyDatasheet

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BiologicalActivity

CompoundLibraries

TechnicalData

SolubilityData

PreparingStockSolutions

MolarityCalculator

ReconstitutionCalculator

DilutionCalculator

ProductDatasheets