Tocris/AQ-RA 741/2292/10/10 mg-免疫在线蚂蚁淘旗下平台

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商品详细Tocris/AQ-RA 741/2292/10/10 mg

Tocris/AQ-RA 741/2292/10/10 mg

商品编号： 2292/10

品牌： Tocris Bioscience

市场价： ¥2980.00

美元价： 1788.00

产地：美国(厂家直采)

公司：

产品分类：受体

公司分类： Receptors

联系Q Q： 3392242852

电话号码： 4000-520-616

电子邮箱： info@ebiomall.com

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商品介绍

Description:Selective,highaffinityM₂antagoNIST

ChemicalName:11-[[4-[4-(Diethylamino)butyl]-1-piperidinyl]acetyl]-5,11-dihydro-6H-pyrido[2,3-b][1,4]benzodiazepin-6-one

Purity:≥99%(HPLC)

BIOLOGicalActivityTechnicalDataSolubilityCalculatorsDatasheetsReferences

BiologicalActivity

Highaffinity,selectivemuscarinicM₂receptorantagonist(pK_ivaluesare8.3,7.7and6.82forM₂,M₁andM₃receptors,respectively).Displayscardioselectivityinvivo,overintestinal,trachealandbladdermuscarinicreceptors;inhibitsvagallyandagonist-inducedbradycardia.

CompoundLibraries

AQ-RA741isalsoofferedaspartoftheTocriscreenPlus.FindoutmoreaboutcompoundlibrariesavailablefromTocris.

TechnicalData

M.Wt	463.62
Formula	C₂₇H₃₇N₅O₂
Storage	StoreatRT
Purity	≥99%(HPLC)
CASNumber	123548-16-3
PubChemID	129989
InChIKey	BCUGCHZRMKTPMU-UHFFFAOYSA-N
Smiles	CCN(CC)CCCCC1CCN(CC(=O)N2C3=CC=CC=C3C(=O)NC3=C2N=CC=C3)CC1

Thetechnicaldataprovidedaboveisforguidanceonly.ForbatchspecificdatarefertotheCertificateofAnalysis.

AllTocrisproductsareintendedforlaboratoryresearchuseonly.

SolubilityData

	Solvent	MaxConc.mg/mL	MaxConc.mM
Solubility
	1eq.HCl	46.36	100
	DMSO	46.36	100
	ethanol	46.36	100

PreparingStockSolutions

Thefollowingdataisbasedontheproductmolecularweight463.62.Batchspecificmolecularweightsmayvaryfrombatchtobatchduetosolventofhydration,whichwillaffectthesolventvolumesrequiredtopreparestocksolutions.

Concentration/SolventVolume/Mass	1mg	5mg	10mg
1mM	2.16mL	10.78mL	21.57mL
5mM	0.43mL	2.16mL	4.31mL
10mM	0.22mL	1.08mL	2.16mL
50mM	0.04mL	0.22mL	0.43mL

ProductDatasheets

CertificateofAnalysis/ProductDatasheet

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BiologicalActivity

CompoundLibraries

TechnicalData

SolubilityData

PreparingStockSolutions

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