BiologicalActivity
5-HT2C/2Breceptoragonist/partialagonist;displayssomeactivityat5-HT2Aand5-HT1receptors.pEC50valuesare7.09,7.2,6.65,5.9and6.5forhumanrecombinant5-HT2C,2Band2A,bovine5-HT1Aandrat5-HT1Breceptorsrespectively.Suppresseslocomotoractivityinratsinvivo.
TechnicalData
M.Wt | 233.14 |
Formula | C10H13ClN2.HCl |
Storage | StoreatRT |
Purity | ≥99%(HPLC) |
CASNumber | 13078-15-4 |
PubChemID | 25681 |
InChIKey | MHXPYWFZULXYHT-UHFFFAOYSA-N |
Smiles | Cl.ClC1=CC=CC(=C1)N1CCNCC1 |
Thetechnicaldataprovidedaboveisforguidanceonly.ForbatchspecificdatarefertotheCertificateofAnalysis.
AllTocrisproductsareintendedforlaboratoryresearchuseonly.
SolubilityData
Solubility | Solubleto100mMinwater |
PreparingStockSolutions
Thefollowingdataisbasedontheproductmolecularweight233.14.Batchspecificmolecularweightsmayvaryfrombatchtobatchduetosolventofhydration,whichwillaffectthesolventvolumesrequiredtopreparestocksolutions.
Concentration/SolventVolume/Mass | 1mg | 5mg | 10mg |
---|---|---|---|
1mM | 4.29mL | 21.45mL | 42.89mL |
5mM | 0.86mL | 4.29mL | 8.58mL |
10mM | 0.43mL | 2.14mL | 4.29mL |
50mM | 0.09mL | 0.43mL | 0.86mL |
MolarityCalculator
ReconstitutionCalculator
Thereconstitutioncalculatorallowsyoutoquicklycalculatethevolumeofareagenttoreconstituteyourvial.Simplyenterthemassofreagentandthetargetconcentrationandthecalculatorwilldeterminetherest.