BiologicalActivity
Anandamidemembranetransportinhibitor(IC50=14μM)thatisrelativelymetabolicallystable.DisplayssomeaffinityforCB2receptorsbuthasonlyweakaffinityforCB1receptorsandhasnoactivityatVR1receptorsorFAAH.AnticonvulsiveinvivofollowingsystemicadmiNISTration.
TechnicalData
| M.Wt | 370.57 |
| Formula | C25H38O2 |
| Storage | Desiccateat-20°C |
| CASNumber | 97452-63-6 |
| PubChemID | 126670 |
| InChIKey | MPJURNPNPDQYSY-LEWJYISDSA-N |
| Smiles | C=[C@](C)[C@@H]1CCC(C)=C[C@H]1[C@]2=C(O)C=C(C(C)(C)CCCCCC)C=C2O |
Thetechnicaldataprovidedaboveisforguidanceonly.ForbatchspecificdatarefertotheCertificateofAnalysis.
AllTocrisproductsareintendedforlaboratoryresearchuseonly.
SolubilityData
| Solubility | Solubleinethanol(suppliedpre-dissolvedinanhydrousethanol,5mg/ml) |
PreparingStockSolutions
Thefollowingdataisbasedontheproductmolecularweight370.57.Batchspecificmolecularweightsmayvaryfrombatchtobatchduetosolventofhydration,whichwillaffectthesolventvolumesrequiredtopreparestocksolutions.
| Concentration/SolventVolume/Mass | 1mg | 5mg | 10mg |
|---|---|---|---|
| 1mM | 2.7mL | 13.49mL | 26.99mL |
| 5mM | 0.54mL | 2.7mL | 5.4mL |
| 10mM | 0.27mL | 1.35mL | 2.7mL |
| 50mM | 0.05mL | 0.27mL | 0.54mL |
MolarityCalculator
ReconstitutionCalculator
Thereconstitutioncalculatorallowsyoutoquicklycalculatethevolumeofareagenttoreconstituteyourvial.Simplyenterthemassofreagentandthetargetconcentrationandthecalculatorwilldeterminetherest.