Tocris/DG 041/6240/10/10毫克
商品编号：
6240
市场价：
¥3580.00
美元价：
2148.00
产品分类：
其他试剂
公司分类：
Other_reagents
联系Q Q：
3392242852
电话号码：
4000-520-616
电子邮箱：
info@ebiomall.com
商品介绍
Description:PotentandselectiveEP3antagoNIST;antiplateletandantithrombotic
ChemicalName:(2E)-3-[1-[(2,4-Dichlorophenyl)methyl]-5-fluoro-3-methyl-1H-indol-7-yl]-N-[(4,5-dichloro-2-thienyl)sulfonyl]-2-propenamide
Purity:≥98%(HPLC)
BIOLOGicalActivityTechnicalDataSolubilityCalculatorsDatasheetsReferences
BiologicalActivity
PotentandselectiveEP3antagonist(IC50=4.6nM).InhibitsPGE2facilitationofplateletaggregationinvitroandexvivo.DisplaysgoodplasmaandmetabolicstABIlity.Doesnotaffectbleedingtimeinrats.Antiplateletandantithrombotic.
TechnicalData
| M.Wt | 592.32 |
| Formula | C23H15Cl4FN2O3S2 |
| Storage | Storeat+4°C |
| Purity | ≥98%(HPLC) |
| CASNumber | 861238-35-9 |
| PubChemID | 11296282 |
| InChIKey | BFBTVZNKWXWKNZ-HWKANZROSA-N |
| Smiles | CC1=CN(C2=C(C=C(C=C12)F)/C=C/C(NS(=O)(C3=CC(Cl)=C(S3)Cl)=O)=O)CC4=C(C=C(C=C4)Cl)Cl |
Thetechnicaldataprovidedaboveisforguidanceonly.ForbatchspecificdatarefertotheCertificateofAnalysis.
AllTocrisproductsareintendedforlaboratoryresearchuseonly.
SolubilityData
| Solvent | MaxConc.mg/mL | MaxConc.mM | |
|---|---|---|---|
| Solubility | |||
| DMSO | 59.23 | 100 |
PreparingStockSolutions
Thefollowingdataisbasedontheproductmolecularweight592.32.Batchspecificmolecularweightsmayvaryfrombatchtobatchduetosolventofhydration,whichwillaffectthesolventvolumesrequiredtopreparestocksolutions.
| Concentration/SolventVolume/Mass | 1mg | 5mg | 10mg |
|---|---|---|---|
| 1mM | 1.69mL | 8.44mL | 16.88mL |
| 5mM | 0.34mL | 1.69mL | 3.38mL |
| 10mM | 0.17mL | 0.84mL | 1.69mL |
| 50mM | 0.03mL | 0.17mL | 0.34mL |
MolarityCalculator
MolarityCalculator
Calculatethemass,volume,orconcentrationrequiredforasolution.
ReconstitutionCalculator
ReconstitutionCalculator
Thereconstitutioncalculatorallowsyoutoquicklycalculatethevolumeofareagenttoreconstituteyourvial.Simplyenterthemassofreagentandthetargetconcentrationandthecalculatorwilldeterminetherest.