Tocris/BGC 20-1531 hydrochloride/5327/10/10 mg-免疫在线蚂蚁淘旗下平台

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商品详细Tocris/BGC 20-1531 hydrochloride/5327/10/10 mg

Tocris/BGC 20-1531 hydrochloride/5327/10/10 mg

商品编号： 5327/10

品牌： Tocris Bioscience

市场价： ¥5980.00

美元价： 3588.00

产地：美国(厂家直采)

公司：

产品分类：受体

公司分类： Receptors

联系Q Q： 3392242852

电话号码： 4000-520-616

电子邮箱： info@ebiomall.com

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商品介绍

Description:HighaffinityandselectiveEP₄antagoNIST

AlternativeNames:PGN1531

ChemicalName:4-[[4-(5-Methoxy-2-pyridinyl)phenoxy]methyl]-5-methyl-N-[(2-methylphenyl)sulfonyl]-2-furancarboxamidehydrochloride

Purity:≥98%(HPLC)

BIOLOGicalActivityTechnicalDataSolubilityCalculatorsDatasheetsReferences

BiologicalActivity

HighaffinityandselectiveEP₄antagonist(K_i=3nM).Exhibits>2500-foldselectivityforEP₄overEP₂andEP₃.Alsoselectiveoverarangeofotherprostanoidreceptors,ionchannels,transportersandenzymes.InhibitsPGE₂-inducedvasodilationofmiddlecerebralandmeningealarteriesinvitro,andcarotidbloodflowinvivo.Orallybioavailable.

TechnicalData

M.Wt	529
Formula	C₂₆H₂₄N₂O₆S.HCl
Storage	DesiccateatRT
Purity	≥98%(HPLC)
PubChemID	121513858
InChIKey	ZSHYZCXOFPPBMH-UHFFFAOYSA-N
Smiles	CC(OC(C(NS(C4=CC=CC=C4C)(=O)=O)=O)=C3)=C3COC(C=C2)=CC=C2C1=NC=C(OC)C=C1.Cl

Thetechnicaldataprovidedaboveisforguidanceonly.ForbatchspecificdatarefertotheCertificateofAnalysis.

AllTocrisproductsareintendedforlaboratoryresearchuseonly.

SolubilityData

	Solvent	MaxConc.mg/mL	MaxConc.mM
Solubility
Solubility	DMSO	49.25	100

PreparingStockSolutions

Thefollowingdataisbasedontheproductmolecularweight529.Batchspecificmolecularweightsmayvaryfrombatchtobatchduetosolventofhydration,whichwillaffectthesolventvolumesrequiredtopreparestocksolutions.

Concentration/SolventVolume/Mass	1mg	5mg	10mg
1mM	1.89mL	9.45mL	18.9mL
5mM	0.38mL	1.89mL	3.78mL
10mM	0.19mL	0.95mL	1.89mL
50mM	0.04mL	0.19mL	0.38mL

ProductDatasheets

CertificateofAnalysis/ProductDatasheet

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