Tocris/BRL 54443/1129/50/50毫克-免疫在线蚂蚁淘旗下平台

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商品详细Tocris/BRL 54443/1129/50/50毫克

Tocris/BRL 54443/1129/50/50毫克

商品编号： 1129/50

品牌： Tocris Bioscience

市场价： ¥10500.00

美元价： 6300.00

产地：美国(厂家直采)

公司：

产品分类：受体

公司分类： Receptors

联系Q Q： 3392242852

电话号码： 4000-520-616

电子邮箱： info@ebiomall.com

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商品介绍

Description:Potent5-ht_1E/FagoNIST

ChemicalName:5-Hydroxy-3-(1-methylpiperidin-4-yl)-1H-indole

BIOLOGicalActivityTechnicalDataSolubilityCalculatorsDatasheetsReferences

BiologicalActivity

Apotent5-ht_1E/1Freceptoragonist(pEC₅₀valuesare8.5and8.6respectively).Displays>30-foldselectivityoverother5-HTanddopaminereceptors(pK_ivaluesare8.7.8.9,7.2,6.9,7.2,5.9,7.0,6.5,<6,<6,6.3and6.2forhuman5-HT_1E,_1F,_1A,_1B,_1D,_2A,_2B,_2C,₄,₇,D₂andD₃receptorsrespectively).Induces5-HT_2Areceptor-mediatedmouseaorticcontractioninvitro(pEC₅₀=6.52).Activeinvivo.

TechnicalData

M.Wt	230.31
Formula	C₁₄H₁₈N₂O
Storage	Desiccateat+4°C
CASNumber	57477-39-1
PubChemID	2438
InChIKey	WKNFADCGOAHBPG-UHFFFAOYSA-N
Smiles	CN1CCC(CC1)C1=CNC2=CC=C(O)C=C12

Thetechnicaldataprovidedaboveisforguidanceonly.ForbatchspecificdatarefertotheCertificateofAnalysis.

AllTocrisproductsareintendedforlaboratoryresearchuseonly.

SolubilityData

Solubility	Solubleto50mMinDMSO

Solubility

Solubleto50mMinDMSO

PreparingStockSolutions

Thefollowingdataisbasedontheproductmolecularweight230.31.Batchspecificmolecularweightsmayvaryfrombatchtobatchduetosolventofhydration,whichwillaffectthesolventvolumesrequiredtopreparestocksolutions.

Concentration/SolventVolume/Mass	1mg	5mg	10mg
1mM	4.34mL	21.71mL	43.42mL
5mM	0.87mL	4.34mL	8.68mL
10mM	0.43mL	2.17mL	4.34mL
50mM	0.09mL	0.43mL	0.87mL

ProductDatasheets

CertificateofAnalysis/ProductDatasheet

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BiologicalActivity

TechnicalData

SolubilityData

PreparingStockSolutions

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