托克里斯/波生坦/6232/50/50毫克-免疫在线蚂蚁淘旗下平台

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商品详细托克里斯/波生坦/6232/50/50毫克

托克里斯/波生坦/6232/50/50毫克

商品编号： 6232/50

品牌： Tocris Bioscience

市场价： ¥5500.00

美元价： 3300.00

产地：美国(厂家直采)

公司：

产品分类：受体

公司分类： Receptors

联系Q Q： 3392242852

电话号码： 4000-520-616

电子邮箱： info@ebiomall.com

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商品介绍

Description:HighaffinitydualET_AandET_BreceptorantagoNIST;orallybioavailable

AlternativeNames:Ro47-0203

ChemicalName:4-(1,1-Dimethylethyl)-N-[6-(2-hydroxyethoxy)-5-(2-methoxyphenoxy)[2,2'-bipyrimidin]-4-yl]benzenesulfonamide

Purity:≥98%(HPLC)

BIOLOGicalActivityTechnicalDataSolubilityCalculatorsDatasheetsReferences

BiologicalActivity

HighaffinitydualET_AandET_Breceptorantagonist(K_ivaluesare4.7and95nMforET_AandET_B,respectively).InhibitsET-1inducedcontractionofisolatedrataortaandsarafotoxinS6C-inducedcontractionofrattracheainvitro.Orallybioavailable.

CompoundLibraries

BosentanisalsoofferedaspartoftheTocriscreenPlus.FindoutmoreaboutcompoundlibrariesavailablefromTocris.

TechnicalData

M.Wt	551.61
Formula	C₂₇H₂₉N₅O₆S
Storage	Storeat+4°C
Purity	≥98%(HPLC)
CASNumber	147536-97-8
PubChemID	104865
InChIKey	GJPICJJJRGTNOD-UHFFFAOYSA-N
Smiles	COC1=C(C=CC=C1)OC2=C(N=C(C3=NC=CC=N3)N=C2NS(=O)(C4=CC=C(C(C)(C)C)C=C4)=O)OCCO

Thetechnicaldataprovidedaboveisforguidanceonly.ForbatchspecificdatarefertotheCertificateofAnalysis.

AllTocrisproductsareintendedforlaboratoryresearchuseonly.

SolubilityData

	Solvent	MaxConc.mg/mL	MaxConc.mM
Solubility
	DMSO	55.16	100
	ethanol	27.58	50

PreparingStockSolutions

Thefollowingdataisbasedontheproductmolecularweight551.61.Batchspecificmolecularweightsmayvaryfrombatchtobatchduetosolventofhydration,whichwillaffectthesolventvolumesrequiredtopreparestocksolutions.

Concentration/SolventVolume/Mass	1mg	5mg	10mg
1mM	1.81mL	9.06mL	18.13mL
5mM	0.36mL	1.81mL	3.63mL
10mM	0.18mL	0.91mL	1.81mL
50mM	0.04mL	0.18mL	0.36mL

ProductDatasheets

CertificateofAnalysis/ProductDatasheet

SafetyDatasheet

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BiologicalActivity

CompoundLibraries

TechnicalData

SolubilityData

PreparingStockSolutions

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ProductDatasheets