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Tocris Bioscience(优势品牌)
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当前位置: 首页 > 产品中心 > Receptors > Tocris/CI 1020/2942/10/10 mg
商品详细Tocris/CI 1020/2942/10/10 mg
Tocris/CI 1020/2942/10/10 mg
Tocris/CI 1020/2942/10/10 mg
商品编号: 2942/10
品牌: Tocris Bioscience
市场价: ¥3780.00
美元价: 2268.00
产地: 美国(厂家直采)
公司:
产品分类: 受体
公司分类: Receptors
联系Q Q: 3392242852
电话号码: 4000-520-616
电子邮箱: info@ebiomall.com
商品介绍
Description:Highlyselective,orallyactiveETAantagoNIST
AlternativeNames:PD156707
ChemicalName:3-(1,3-Benzodioxol-5-yl)-5-hydroxy-5-(4-methoxyphenyl)-4-[(3,4,5-trimethoxyphenyl)methyl]-2(5H)-furanone
Purity:≥98%(HPLC)
BIOLOGicalActivityTechnicalDataSolubilityCalculatorsDatasheetsReferences

BiologicalActivity

Highlyselective,orallyactive,non-peptideendothelin-Areceptor(ETA)antagonist(IC50valuesare0.3and480nMforETAandETBreceptorsrespectively).Antihypertensive;blocksET-1-inducedpressorresponsesfollowingoraladministration.

LicensingInformation

SoldforresearchpurposesunderagreementfromPfizerInc.

TechnicalData

M.Wt506.5
FormulaC28H26O9
StorageStoreat-20°C
Purity≥98%(HPLC)
CASNumber162256-50-0
PubChemID9870830
InChIKeyPWIPORDFWDZCJG-UHFFFAOYSA-N
SmilesO=C1C(C2=CC=C(OCO4)C4=C2)=C(CC3=CC(OC)=C(OC)C(OC)=C3)C(O)(C5=CC=C(OC)C=C5)O1

Thetechnicaldataprovidedaboveisforguidanceonly.ForbatchspecificdatarefertotheCertificateofAnalysis.

AllTocrisproductsareintendedforlaboratoryresearchuseonly.

SolubilityData

SolventMaxConc.mg/mLMaxConc.mM
Solubility
DMSO25.3250

PreparingStockSolutions

Thefollowingdataisbasedontheproductmolecularweight506.5.Batchspecificmolecularweightsmayvaryfrombatchtobatchduetosolventofhydration,whichwillaffectthesolventvolumesrequiredtopreparestocksolutions.

Concentration/SolventVolume/Mass1mg5mg10mg
1mM1.97mL9.87mL19.74mL
5mM0.39mL1.97mL3.95mL
10mM0.2mL0.99mL1.97mL
50mM0.04mL0.2mL0.39mL

ProductDatasheets

CertificateofAnalysis/ProductDatasheet
SafetyDatasheet