Tocris/CI 988/2607/50/50 mg-免疫在线蚂蚁淘旗下平台

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商品详细Tocris/CI 988/2607/50/50 mg

Tocris/CI 988/2607/50/50 mg

商品编号： 2607/50

品牌： Tocris Bioscience

市场价： ¥22100.00

美元价： 13260.00

产地：美国(厂家直采)

公司：

产品分类：受体

公司分类： Receptors

联系Q Q： 3392242852

电话号码： 4000-520-616

电子邮箱： info@ebiomall.com

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商品介绍

Description:PotentandselectiveCCK₂antagoNIST

AlternativeNames:PD134308

ChemicalName:4-[[(1R)-2-[[(2R)-3-(1H-indol-3-yl)-2-methyl-1-oxo-2-[[(tricyclo[3.3.1.13,7]dec-2-yloxy)carbonyl]amino]propyl]amino]-1-phenylethyl]amino]-4-oxobutanoicacid

Purity:≥99%(HPLC)

BIOLOGicalActivityTechnicalDataSolubilityCalculatorsDatasheetsReferences

BiologicalActivity

PotentandselectiveCCK₂(CCK-B)receptorantagonistthatdisplays~1600-foldselectivityoverCCK₁receptors(IC₅₀valuesare1.7and2717nMforCCK₂andCCK₁respectively).HasnegligIBLeaffinityatarangeofotherbindingsites(IC₅₀>10μM).Exhibitsanxiolyticactivityfollowingoraladministration.

TechnicalData

M.Wt	614.73
Formula	C₃₅H₄₂N₄O₆
Storage	Storeat+4°C
Purity	≥99%(HPLC)
CASNumber	130332-27-3
PubChemID	108187
InChIKey	FVQSSYMRZKLFDR-ZABPBAJSSA-N
Smiles	C[C@](NC(OC5C3CC(CC5C6)CC6C3)=O)(C(NC[C@@H]([C@]4=CC=CC=C4)NC(CCC(O)=O)=O)=O)CC2=CNC1=CC=CC=C12

Thetechnicaldataprovidedaboveisforguidanceonly.ForbatchspecificdatarefertotheCertificateofAnalysis.

AllTocrisproductsareintendedforlaboratoryresearchuseonly.

SolubilityData

	Solvent	MaxConc.mg/mL	MaxConc.mM
Solubility
Solubility	DMSO	61.47	100

PreparingStockSolutions

Thefollowingdataisbasedontheproductmolecularweight614.73.Batchspecificmolecularweightsmayvaryfrombatchtobatchduetosolventofhydration,whichwillaffectthesolventvolumesrequiredtopreparestocksolutions.

Concentration/SolventVolume/Mass	1mg	5mg	10mg
1mM	1.63mL	8.13mL	16.27mL
5mM	0.33mL	1.63mL	3.25mL
10mM	0.16mL	0.81mL	1.63mL
50mM	0.03mL	0.16mL	0.33mL

ProductDatasheets

CertificateofAnalysis/ProductDatasheet

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BiologicalActivity

TechnicalData

SolubilityData

PreparingStockSolutions

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