Biological Activity
5-HT2 antagonist.
Technical Data
| M. Wt | 376.94 |
| Formula | C20H24N2OS.HCl |
| Storage | Desiccate at RT |
| Purity | ≥99% (HPLC) |
| CAS Number | 54-84-2 |
| PubChem ID | 6433141 |
| InChI Key | LXGJPDKYMJJWRB-IERUDJENSA-N |
| Smiles | O=C(/C=C/C2=CC=CC=C2)NC1=CC=CC=C1SCCCN(C)C.Cl |
The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
All Tocris products are intended for laboratory research use only.
Solubility Data
| Solubility | Soluble to 50 mM in water |
Preparing Stock Solutions
The following data is based on the product molecular weight 376.94. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.
| Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
|---|---|---|---|
| 1 mM | 2.65 mL | 13.26 mL | 26.53 mL |
| 5 mM | 0.53 mL | 2.65 mL | 5.31 mL |
| 10 mM | 0.27 mL | 1.33 mL | 2.65 mL |
| 50 mM | 0.05 mL | 0.27 mL | 0.53 mL |
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Product Datasheets
References
References are publications that support the products' biological activity.
Leysen et al (1981) Receptor binding profile of R-41-468, a novel antagonist at 5HT2 receptors. Life Sci. 28 1015 PMID: 6261070
Pierce et al (1992) Molecular structure basis of ligand selectivity for 5-HT2 versus 5-HT1C cortical receptors. Naunyn Schmiedebergs Arch.Pharmacol. 346 4 PMID: 1407003
Keywords: Cinanserin hydrochloride, supplier, Selective, 5-HT2, antagonists, Non-Selective, Serotonin, Receptors, Non-selective, 5-HT2, Non-selective, 5-HT2, Tocris Bioscience
