Tocris/Eplivanserin hemifumarate/4958/10/10 mg-免疫在线蚂蚁淘旗下平台

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商品详细Tocris/Eplivanserin hemifumarate/4958/10/10 mg

Tocris/Eplivanserin hemifumarate/4958/10/10 mg

商品编号： 4958/10

品牌： Tocris Bioscience

市场价： ¥3100.00

美元价： 1860.00

产地：美国(厂家直采)

公司：

产品分类：受体

公司分类： Receptors

联系Q Q： 3392242852

电话号码： 4000-520-616

电子邮箱： info@ebiomall.com

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商品介绍

Description:Potentandselective5-HT_2AantagoNIST

AlternativeNames:SR-46349hemifumarate,SR-46349B

ChemicalName:(1Z,2E)-1-(2-Fluorophenyl)-3-(4-hydroxyphenyl)-2-propen-1-oneO-[2-(dimethylamino)ethyl]oximehemifumarate

Purity:≥98%(HPLC)

BIOLOGicalActivityTechnicalDataSolubilityCalculatorsDatasheetsReferences

BiologicalActivity

Potentandselective5-HT_2Aantagonist(IC₅₀valuesare5.8and120and>100nMfor5-HT_2A,5-HT_2Band5-HT_2C,respectively).Attenuatescocaine-inducedhyperactivity.Increasesdopamine(DA)releaseinratmedialprefrontalcortex(mPFC);potentiateshaloperidol-inducedDAreleaseinthemPFCandnucleusaccumbens.

TechnicalData

M.Wt	386.42
Formula	C₁₉H₂₁FN₂O₂.0.5C₄H₄O₄
Storage	Storeat+4°C
Purity	≥98%(HPLC)
CASNumber	130580-02-8
PubChemID	6438382
InChIKey	UCLIFEBROADCQW-PWERMGERSA-N
Smiles	OC(C=C2)=CC=C2/C=C/C(C1=CC=CC=C1F)=N/OCCN(C)C.O=C(/C=C/C(O)=O)O.OC(C=C4)=CC=C4/C=C/C(C3=CC=CC=C3F)=N/OCCN(C)C

Thetechnicaldataprovidedaboveisforguidanceonly.ForbatchspecificdatarefertotheCertificateofAnalysis.

AllTocrisproductsareintendedforlaboratoryresearchuseonly.

SolubilityData

	Solvent	MaxConc.mg/mL	MaxConc.mM
Solubility
Solubility	DMSO	19.32	50

PreparingStockSolutions

Thefollowingdataisbasedontheproductmolecularweight386.42.Batchspecificmolecularweightsmayvaryfrombatchtobatchduetosolventofhydration,whichwillaffectthesolventvolumesrequiredtopreparestocksolutions.

Concentration/SolventVolume/Mass	1mg	5mg	10mg
1mM	2.59mL	12.94mL	25.88mL
5mM	0.52mL	2.59mL	5.18mL
10mM	0.26mL	1.29mL	2.59mL
50mM	0.05mL	0.26mL	0.52mL

ProductDatasheets

CertificateofAnalysis/ProductDatasheet

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BiologicalActivity

TechnicalData

SolubilityData

PreparingStockSolutions

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