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商品详细Tocris/G-15/3678/10/10毫克

Tocris/G-15/3678/10/10毫克

商品编号： 3678/10

品牌： Tocris Bioscience

市场价： ¥3780.00

美元价： 2268.00

产地：美国(厂家直采)

公司：

产品分类：受体

公司分类： Receptors

联系Q Q： 3392242852

电话号码： 4000-520-616

电子邮箱： info@ebiomall.com

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商品介绍

Description:HighaffinityandselectiveGPERantagoNIST

ChemicalName:(3aS*,4R*,9bR*)-4-(6-Bromo-1,3-benzodioxol-5-yl)-3a,4,5,9b-3H-cyclopenta[c]quinoline

Purity:≥99%(HPLC)

BIOLOGicalActivityTechnicalDataSolubilityCalculatorsDatasheetsReferences

BiologicalActivity

HighaffinityandselectiveGPERreceptorantagonist(K_i=20nM)thatdisplaysnoaffinityforERαandERβatconcentrationsupto10μM.Inhibitsagonist-inducedcalciummobilizationinvitro(EC₅₀of~185nM)andantagonizestheantidepressiveandrenoprotectiveeffectsofestrogeninvivo.

TechnicalData

M.Wt	370.24
Formula	C₁₉H₁₆BrNO₂
Storage	Storeat-20°C
Purity	≥99%(HPLC)
CASNumber	1161002-05-6
PubChemID	90488870
InChIKey	LBBDCJLRQXMUAE-FWHYVADDSA-N
Smiles	BrC1=CC4=C(OCO4)C=[C@@]1[C@@H]2NC(C=CC=C5)=C5[C@@]3([H])[C@@]([H])2CC=C3.BrC6=CC9=C(OCO9)C=[C@@]6[C@H]7NC(C=CC=C%10)=C%10[C@]8([H])[C@]([H])7CC=C8

Thetechnicaldataprovidedaboveisforguidanceonly.ForbatchspecificdatarefertotheCertificateofAnalysis.

AllTocrisproductsareintendedforlaboratoryresearchuseonly.

SolubilityData

	Solvent	MaxConc.mg/mL	MaxConc.mM
Solubility
Solubility	DMSO	18.51	50

PreparingStockSolutions

Thefollowingdataisbasedontheproductmolecularweight370.24.Batchspecificmolecularweightsmayvaryfrombatchtobatchduetosolventofhydration,whichwillaffectthesolventvolumesrequiredtopreparestocksolutions.

Concentration/SolventVolume/Mass	1mg	5mg	10mg
1mM	2.7mL	13.5mL	27.01mL
5mM	0.54mL	2.7mL	5.4mL
10mM	0.27mL	1.35mL	2.7mL
50mM	0.05mL	0.27mL	0.54mL

ProductDatasheets

CertificateofAnalysis/ProductDatasheet

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BiologicalActivity

TechnicalData

SolubilityData

PreparingStockSolutions

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