Tocris/GNTI dihydrochloride/1282/10/10 mg-免疫在线蚂蚁淘旗下平台

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商品详细Tocris/GNTI dihydrochloride/1282/10/10 mg

Tocris/GNTI dihydrochloride/1282/10/10 mg

商品编号： 1282/10

品牌： Tocris Bioscience

市场价： ¥3980.00

美元价： 2388.00

产地：美国(厂家直采)

公司：

产品分类：受体

公司分类： Receptors

联系Q Q： 3392242852

电话号码： 4000-520-616

电子邮箱： info@ebiomall.com

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商品介绍

Description:Potent,selectiveκantagoNIST

ChemicalName:5'-Guanidinyl-17-(cyclopropylmethyl)-6,7-dehydro-4,5α-epoxy-3,14-dihydroxy-6,7-2',3'-indolomorphinandihydrochloride

Purity:≥96%(HPLC)

BIOLOGicalActivityTechnicalDataSolubilityCalculatorsDatasheetsReferences

BiologicalActivity

Highlypotentκopioidreceptorantagonist(K_i=0.18nMforhumanclonedκreceptorsexpressedinCHOcells).Displays208-and799-foldselectivityoverμandδreceptorsrespectively.Reducesfeedingbehaviorinratswithamuchhigherpotency(300-30,000-fold)andashorterdurationofactionthannor-binaltorphimine(Cat.No.0347).

TechnicalData

M.Wt	544.48
Formula	C₂₇H₂₉N₅O₃.2HCl
Storage	Desiccateat-20°C
Purity	≥96%(HPLC)
CASNumber	351183-88-5
PubChemID	90479777
InChIKey	GJPIMNXJPMPQHK-CVVXFVLRSA-N
Smiles	OC3=CC=C2CC([C@@]5(O)[C@@]4(CC8)C2=C3O[C@H]4C(NC7=C6C=C(NC=N)C=C7)=C6C5)N8CC1CC1.Cl.Cl

Thetechnicaldataprovidedaboveisforguidanceonly.ForbatchspecificdatarefertotheCertificateofAnalysis.

AllTocrisproductsareintendedforlaboratoryresearchuseonly.

SolubilityData

	Solvent	MaxConc.mg/mL	MaxConc.mM
Solubility
	DMSO	54.45	100
	water	54.45	100

PreparingStockSolutions

Thefollowingdataisbasedontheproductmolecularweight544.48.Batchspecificmolecularweightsmayvaryfrombatchtobatchduetosolventofhydration,whichwillaffectthesolventvolumesrequiredtopreparestocksolutions.

Concentration/SolventVolume/Mass	1mg	5mg	10mg
1mM	1.84mL	9.18mL	18.37mL
5mM	0.37mL	1.84mL	3.67mL
10mM	0.18mL	0.92mL	1.84mL
50mM	0.04mL	0.18mL	0.37mL

ProductDatasheets

CertificateofAnalysis/ProductDatasheet

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TechnicalData

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