Tocris/GR 125487 sulfamate/1658/10/10 mg-免疫在线蚂蚁淘旗下平台

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商品详细Tocris/GR 125487 sulfamate/1658/10/10 mg

Tocris/GR 125487 sulfamate/1658/10/10 mg

商品编号： 1658/10

品牌： Tocris Bioscience

市场价： ¥3780.00

美元价： 2268.00

产地：美国(厂家直采)

公司：

产品分类：受体

公司分类： Receptors

联系Q Q： 3392242852

电话号码： 4000-520-616

电子邮箱： info@ebiomall.com

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商品介绍

Description:Potent,selective5-HT₄antagoNIST;activeinvivo

ChemicalName:5-Fluoro-2-methoxy-[1-[2-[(methylsulfonyl)amino]ethyl]-4-piperidinyl]-1H-indole-3-methylcarboxylatesulfamate

Purity:≥97%(HPLC)

BIOLOGicalActivityTechnicalDataSolubilityCalculatorsDatasheetsReferences

BiologicalActivity

Potentandselective5-HT₄receptorantagonist(K_i=0.19nMforporcine5-HT₄).Centrallyactivefollowingsystemicadministrationinvivo.

LicensingInformation

SoldforresearchpurposesunderagreementfromGlaxoSmithKline

TechnicalData

M.Wt	524.58
Formula	C₁₉H₂₆FN₃O₅S.H₂NSO₃H
Storage	DesiccateatRT
Purity	≥97%(HPLC)
CASNumber	859502-43-5
PubChemID	6604955
InChIKey	VQJFDBXITIOGJM-UHFFFAOYSA-N
Smiles	NS(O)(=O)=O.COC1=C(C(=O)OCC2CCN(CCNS(C)(=O)=O)CC2)C2=CC(F)=CC=C2N1

Thetechnicaldataprovidedaboveisforguidanceonly.ForbatchspecificdatarefertotheCertificateofAnalysis.

AllTocrisproductsareintendedforlaboratoryresearchuseonly.

SolubilityData

	Solvent	MaxConc.mg/mL	MaxConc.mM
Solubility
	phosphatebufferedsaline	2.14	5mMwithgentlewarming
	water	4.27	10mMwithgentlewarming

PreparingStockSolutions

Thefollowingdataisbasedontheproductmolecularweight524.58.Batchspecificmolecularweightsmayvaryfrombatchtobatchduetosolventofhydration,whichwillaffectthesolventvolumesrequiredtopreparestocksolutions.

Concentration/SolventVolume/Mass	1mg	5mg	10mg
1mM	1.91mL	9.53mL	19.06mL
5mM	0.38mL	1.91mL	3.81mL
10mM	0.19mL	0.95mL	1.91mL
50mM	0.04mL	0.19mL	0.38mL

ProductDatasheets

CertificateofAnalysis/ProductDatasheet

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BiologicalActivity

LicensingInformation

TechnicalData

SolubilityData

PreparingStockSolutions

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ProductDatasheets