Tocris/GSK LSD 1 dihydrochloride/5361/10/10 mg-免疫在线蚂蚁淘旗下平台

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商品详细Tocris/GSK LSD 1 dihydrochloride/5361/10/10 mg

Tocris/GSK LSD 1 dihydrochloride/5361/10/10 mg

商品编号： 5361/10

品牌： Tocris Bioscience

市场价： ¥3300.00

美元价： 1980.00

产地：美国(厂家直采)

公司：

产品分类：其它酶

公司分类： Other_enzymes

联系Q Q： 3392242852

电话号码： 4000-520-616

电子邮箱： info@ebiomall.com

立即询价

商品介绍

Description:PotentandselectiveLSD1inhibitor

ChemicalName:rel-N-[(1S,2R)-2-Phenylcyclopropyl]-4-piperidinaminedihydrochloride

Purity:≥98%(HPLC)

BIOLOGicalActivityTechnicalDataSolubilityCalculatorsDatasheetsReferences

BiologicalActivity

Potentandselectivelysinespecificdemethylase1(LSD1)inhibitor(IC₅₀=16nM).Exhibits>1000-foldselectivityforLSD1overcloselyrelatedenzymesincludingLSD2,MAO-1andMAO-B.Inhibitscancercelllinegrowthinvitro.

LicensingInformation

ThisprobeissuppliedinconjunctionwiththeStructuralGenomicsConsortium.Forfurthercharacterizationdetails,pleasevisittheGSKLSD1probesummaryontheSGCwebsite.

CompoundLibraries

GSKLSD1dihydrochlorideisalsoofferedaspartoftheTocriscreenPlus.FindoutmoreaboutcompoundlibrariesavailablefromTocris.

TechnicalData

M.Wt	289.24
Formula	C₁₄H₂₀N₂.2HCl
Storage	Storeat+4°C
Purity	≥98%(HPLC)
PubChemID	91663353
InChIKey	PJFZOGMSPBHPNS-WICJZZOFSA-N
Smiles	C1(N[C@@H]2C[C@H]2[C@]3=CC=CC=C3)CCNCC1.Cl.Cl

Thetechnicaldataprovidedaboveisforguidanceonly.ForbatchspecificdatarefertotheCertificateofAnalysis.

AllTocrisproductsareintendedforlaboratoryresearchuseonly.

SolubilityData

	Solvent	MaxConc.mg/mL	MaxConc.mM
Solubility
	DMSO	28.92	100
	water	28.92	100

PreparingStockSolutions

Thefollowingdataisbasedontheproductmolecularweight289.24.Batchspecificmolecularweightsmayvaryfrombatchtobatchduetosolventofhydration,whichwillaffectthesolventvolumesrequiredtopreparestocksolutions.

Concentration/SolventVolume/Mass	1mg	5mg	10mg
1mM	3.46mL	17.29mL	34.57mL
5mM	0.69mL	3.46mL	6.91mL
10mM	0.35mL	1.73mL	3.46mL
50mM	0.07mL	0.35mL	0.69mL

ProductDatasheets

CertificateofAnalysis/ProductDatasheet

SafetyDatasheet

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