Tocris/纳络酮苯甲酰腙/1419/50/50 mg-免疫在线蚂蚁淘旗下平台

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商品详细Tocris/纳络酮苯甲酰腙/1419/50/50 mg

Tocris/纳络酮苯甲酰腙/1419/50/50 mg

商品编号： 1419/50

品牌： Tocris Bioscience

市场价： ¥9700.00

美元价： 5820.00

产地：美国(厂家直采)

公司：

产品分类：受体

公司分类： Receptors

联系Q Q： 3392242852

电话号码： 4000-520-616

电子邮箱： info@ebiomall.com

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商品介绍

Description:FullκagoNIST,partialμandδagonistandantagonizesagonist-inducedactivationofNOP

AlternativeNames:NalBzOH

ChemicalName:[(5α)-4,5-Epoxy-3,14-dihydroxy-17-(2-propenyl)morphinan-6-ylidene]benzoicacidhydrazide

Purity:≥99%(HPLC)

BIOLOGicalActivityTechnicalDataSolubilityCalculatorsDatasheetsReferences

BiologicalActivity

Mixedopioidreceptoragonist/antagonist.Actsasapotentandfullagonistatκ,apartialagonistatμandδopioidreceptors(pEC₅₀valuesare9.45,8.74and8.61inacAMPassay,9.70,8.59and8.49ina[³⁵S]GTPγSbindingassayrespectively).FailstoexertagonisteffectsatNOPreceptorsandantagonizesagonist-inducedNOPactivation.Stimulatesκ-,μ-andδ-mediatedanalgesiaandblocksNOP-inducedsupraspinalnociception.

TechnicalData

M.Wt	445.52
Formula	C₂₆H₂₇N₃O₄
Storage	Desiccateat+4°C
Purity	≥99%(HPLC)
CASNumber	119630-94-3
PubChemID	9601084
InChIKey	AKXCFAYOTIEFOH-XTNAHFASSA-N
Smiles	O[C@@]23[C@@]([C@]5([H])/C(CC3)=N/NC(C6=CC=CC=C6)=O)(CC4)C1=C(O5)C(O)=CC=C1C[C@H]2N4CC=C

Thetechnicaldataprovidedaboveisforguidanceonly.ForbatchspecificdatarefertotheCertificateofAnalysis.

AllTocrisproductsareintendedforlaboratoryresearchuseonly.

SolubilityData

	Solvent	MaxConc.mg/mL	MaxConc.mM
Solubility
Solubility	DMSO	22.28	50

PreparingStockSolutions

Thefollowingdataisbasedontheproductmolecularweight445.52.Batchspecificmolecularweightsmayvaryfrombatchtobatchduetosolventofhydration,whichwillaffectthesolventvolumesrequiredtopreparestocksolutions.

Concentration/SolventVolume/Mass	1mg	5mg	10mg
1mM	2.24mL	11.22mL	22.45mL
5mM	0.45mL	2.24mL	4.49mL
10mM	0.22mL	1.12mL	2.24mL
50mM	0.04mL	0.22mL	0.45mL

ProductDatasheets

CertificateofAnalysis/ProductDatasheet

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BiologicalActivity

TechnicalData

SolubilityData

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