Tocris/WIN 55212-3甲磺酸酯/2327/50/50毫克-免疫在线蚂蚁淘旗下平台

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商品详细Tocris/WIN 55212-3甲磺酸酯/2327/50/50毫克

Tocris/WIN 55212-3甲磺酸酯/2327/50/50毫克

商品编号： 2327/50

品牌： Tocris Bioscience

市场价： ¥10700.00

美元价： 6420.00

产地：美国(厂家直采)

公司：

产品分类：受体

公司分类： Receptors

联系Q Q： 3392242852

电话号码： 4000-520-616

电子邮箱： info@ebiomall.com

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商品介绍

Description:CB₂antagoNIST/CB₁partialinverseagonist;enantiomerofWIN55,212-2(Cat.No.1038)

AlternativeNames:(S)-(-)-WIN55,212

ChemicalName:[(3S)-2,3-Dihydro-5-methyl-3-(4-morpholinylmethyl)pyrrolo[1,2,3-de]-1,4-benzoxazin-6-yl]-1-naphthalenyl-methanonemonomethanesulfonate

Purity:≥98%(HPLC)

BIOLOGicalActivityTechnicalDataSolubilityCalculatorsDatasheetsReferences

BiologicalActivity

Novel,lowpotencyCB₂receptorsilentantagonistandCB₁receptorpartialinverseagonist.CompetitivelyantagonizeseffectsofCP55,940(pA₂=6.1)andSR144528(pEC₅₀=5.3)atCB₂receptorsandactsasapartialinverseagonistatCB₁receptors(pIC₅₀=5.5).DisplaysmodestactivityathumanmelatoninMT₁andmuscarinicM₄receptors,butisselectiveoverseveralotherGPCRs.

TechnicalData

M.Wt	522.61
Formula	C₂₇H₂₆N₂O₃.CH₃SO₃H
Storage	Storeat+4°C
Purity	≥98%(HPLC)
CASNumber	131543-25-4
PubChemID	11613341
InChIKey	FSGCSTPOPBJYSX-BDQAORGHSA-N
Smiles	CS(O)(=O)=O.CC1=C(C(=O)C2=CC=CC3=C2C=CC=C3)C2=CC=CC3=C2N1[C@@H](CN1CCOCC1)CO3

Thetechnicaldataprovidedaboveisforguidanceonly.ForbatchspecificdatarefertotheCertificateofAnalysis.

AllTocrisproductsareintendedforlaboratoryresearchuseonly.

SolubilityData

	Solvent	MaxConc.mg/mL	MaxConc.mM
Solubility
Solubility	DMSO	52.26	100mMwithgentlewarming

PreparingStockSolutions

Thefollowingdataisbasedontheproductmolecularweight522.61.Batchspecificmolecularweightsmayvaryfrombatchtobatchduetosolventofhydration,whichwillaffectthesolventvolumesrequiredtopreparestocksolutions.

Concentration/SolventVolume/Mass	1mg	5mg	10mg
1mM	1.91mL	9.57mL	19.13mL
5mM	0.38mL	1.91mL	3.83mL
10mM	0.19mL	0.96mL	1.91mL
50mM	0.04mL	0.19mL	0.38mL

ProductDatasheets

CertificateofAnalysis/ProductDatasheet

SafetyDatasheet

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BiologicalActivity

TechnicalData

SolubilityData

PreparingStockSolutions

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