Tocris/J 104129 fumarate/2507/10/10 mg-免疫在线蚂蚁淘旗下平台

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商品详细Tocris/J 104129 fumarate/2507/10/10 mg

Tocris/J 104129 fumarate/2507/10/10 mg

商品编号： 2507/10

品牌： Tocris Bioscience

市场价： ¥3780.00

美元价： 2268.00

产地：美国(厂家直采)

公司：

产品分类：受体

公司分类： Receptors

联系Q Q： 3392242852

电话号码： 4000-520-616

电子邮箱： info@ebiomall.com

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商品介绍

Description:Potent,selectiveM₃antagoNIST

ChemicalName:(αR)-α-Cyclopentyl-α-hydroxy-N-[1-(4-methyl-3-pentenyl)-4-piperidinyl]benzeneacetamidefumarate

Purity:≥99%(HPLC)

BIOLOGicalActivityTechnicalDataSolubilityCalculatorsDatasheetsReferences

BiologicalActivity

PotentM₃muscarinicreceptorantagonistthatdisplays~120-foldselectivityoverM₂receptors(K_ivaluesare4.2,19and490nMforhumanM₃,M₁andM₂receptorsrespectively).Exhibits>250-foldbronchialselectivity;inhibitsACh-inducedbronchoconstrictionbutnotACh-inducedbradycardia(K_Bvaluesare3.3and170nMforrattracheaM₃andratrightatriaM₂receptorsrespectively).

TechnicalData

M.Wt	500.63
Formula	C₂₄H₃₆N₂O₂.C₄H₄O₄
Storage	Storeat+4°C
Purity	≥99%(HPLC)
CASNumber	257603-40-0
PubChemID	56972189
InChIKey	HUCQUCITPHOUAC-DSSYAJFBSA-N
Smiles	[H]OC(=O)C=CC(=O)O[H].CC(C)=CCCN1CCC(CC1)NC(=O)[C@@](O)(C1CCCC1)C1=CC=CC=C1

Thetechnicaldataprovidedaboveisforguidanceonly.ForbatchspecificdatarefertotheCertificateofAnalysis.

AllTocrisproductsareintendedforlaboratoryresearchuseonly.

SolubilityData

	Solvent	MaxConc.mg/mL	MaxConc.mM
Solubility
	DMSO	50.06	100
	ethanol	25.03	50

PreparingStockSolutions

Thefollowingdataisbasedontheproductmolecularweight500.63.Batchspecificmolecularweightsmayvaryfrombatchtobatchduetosolventofhydration,whichwillaffectthesolventvolumesrequiredtopreparestocksolutions.

Concentration/SolventVolume/Mass	1mg	5mg	10mg
1mM	2mL	9.99mL	19.97mL
5mM	0.4mL	2mL	3.99mL
10mM	0.2mL	1mL	2mL
50mM	0.04mL	0.2mL	0.4mL

ProductDatasheets

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BiologicalActivity

TechnicalData

SolubilityData

PreparingStockSolutions

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