Tocris/JZP 361/5851/50/50 mg-免疫在线蚂蚁淘旗下平台

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商品详细Tocris/JZP 361/5851/50/50 mg

Tocris/JZP 361/5851/50/50 mg

商品编号： 5851/50

品牌： Tocris Bioscience

市场价： ¥12580.00

美元价： 7548.00

产地：美国(厂家直采)

公司：

产品分类：其它酶

公司分类： Other_enzymes

联系Q Q： 3392242852

电话号码： 4000-520-616

电子邮箱： info@ebiomall.com

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商品介绍

Description:PotentandselectivereversIBLeMAGLinhibitor

ChemicalName:[4-(8-Chloro-5,6-dihydro-11H-benzo[5,6]cyclohepta[1,2-b]pyridin-11-ylidene)-1-piperidinyl](1H-1,2,4-triazol-1-yl)methanone

Purity:≥99%(HPLC)

BIOLOGicalActivityTechnicalDataSolubilityCalculatorsDatasheetsReferences

BiologicalActivity

PotentandselectivereversibleMAGLinhibitor(IC₅₀=46nM).Exhibits35-foldand150-foldhigherselectivityoverhumanFAAHandABHD6,respectively(IC₅₀valuesare1.79and7.24μM,respectively).DisplaysaffinityforH₁receptors(pA₂=6.81).ExhibitsnoactivityatcannABInoidreceptorsat10μM.

TechnicalData

M.Wt	405.88
Formula	C₂₂H₂₀ClN₅O
Storage	Storeat+4°C
Purity	≥99%(HPLC)
CASNumber	1680193-80-9
PubChemID	102596130
InChIKey	GAVZCGTYRWKKDV-UHFFFAOYSA-N
Smiles	ClC1=CC=C2C(CCC3=CC=CN=C3/C2=C4CCN(C(N5C=NC=N5)=O)CC4)=C1

Thetechnicaldataprovidedaboveisforguidanceonly.ForbatchspecificdatarefertotheCertificateofAnalysis.

AllTocrisproductsareintendedforlaboratoryresearchuseonly.

SolubilityData

	Solvent	MaxConc.mg/mL	MaxConc.mM
Solubility
	DMSO	40.59	100
	ethanol	8.12	20

PreparingStockSolutions

Thefollowingdataisbasedontheproductmolecularweight405.88.Batchspecificmolecularweightsmayvaryfrombatchtobatchduetosolventofhydration,whichwillaffectthesolventvolumesrequiredtopreparestocksolutions.

Concentration/SolventVolume/Mass	1mg	5mg	10mg
1mM	2.46mL	12.32mL	24.64mL
5mM	0.49mL	2.46mL	4.93mL
10mM	0.25mL	1.23mL	2.46mL
50mM	0.05mL	0.25mL	0.49mL

ProductDatasheets

CertificateofAnalysis/ProductDatasheet

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BiologicalActivity

TechnicalData

SolubilityData

PreparingStockSolutions

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