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商品详细Tocris/KW 3902/4167/50/50 mg

Tocris/KW 3902/4167/50/50 mg

商品编号： 4167/50

品牌： Tocris Bioscience

市场价： ¥14180.00

美元价： 8508.00

产地：美国(厂家直采)

公司：

产品分类：受体

公司分类： Receptors

联系Q Q： 3392242852

电话号码： 4000-520-616

电子邮箱： info@ebiomall.com

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商品介绍

Description:SelectiveA₁antagoNIST

AlternativeNames:Rolofylline

ChemicalName:8-(Hexahydro-2,5-methanopentalen-3a(1H)-yl)-3,7-dihydro-1,3-dipropyl-1H-purine-2,6-dione

Purity:≥99%(HPLC)

BIOLOGicalActivityTechnicalDataSolubilityCalculatorsDatasheetsReferences

BiologicalActivity

SelectiveadenosineA₁receptorantagonist;displays890-foldselectivityforratA₁receptorsoverA_2Areceptors(K_ivaluesare0.19and170nMrespectively).DisplaysnoeffectonrecombinantratA₃receptorsexpressedonCHOcellsatconcentrationsupto10μM.Exhibitsdiureticandrenalprotectiveeffectsinrats.

CompoundLibraries

KW3902isalsoofferedaspartoftheTocriscreenPlus.FindoutmoreaboutcompoundlibrariesavailablefromTocris.

TechnicalData

M.Wt	356.46
Formula	C₂₀H₂₈N₄O₂
Storage	Storeat+4°C
Purity	≥99%(HPLC)
CASNumber	136199-02-5
PubChemID	64627
InChIKey	PJBFVWGQFLYWCB-UHFFFAOYSA-N
Smiles	O=C1C2=C(NC(C34CC(CC4C5)CC5C3)=N2)N(CCC)C(N1CCC)=O

Thetechnicaldataprovidedaboveisforguidanceonly.ForbatchspecificdatarefertotheCertificateofAnalysis.

AllTocrisproductsareintendedforlaboratoryresearchuseonly.

SolubilityData

	Solvent	MaxConc.mg/mL	MaxConc.mM
Solubility
	DMSO	17.82	50
	ethanol	8.91	25

PreparingStockSolutions

Thefollowingdataisbasedontheproductmolecularweight356.46.Batchspecificmolecularweightsmayvaryfrombatchtobatchduetosolventofhydration,whichwillaffectthesolventvolumesrequiredtopreparestocksolutions.

Concentration/SolventVolume/Mass	1mg	5mg	10mg
1mM	2.81mL	14.03mL	28.05mL
5mM	0.56mL	2.81mL	5.61mL
10mM	0.28mL	1.4mL	2.81mL
50mM	0.06mL	0.28mL	0.56mL

ProductDatasheets

CertificateofAnalysis/ProductDatasheet

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BiologicalActivity

CompoundLibraries

TechnicalData

SolubilityData

PreparingStockSolutions

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