Tocris/LY 2183240/2452/1/1毫克-免疫在线蚂蚁淘旗下平台

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商品详细Tocris/LY 2183240/2452/1/1毫克

Tocris/LY 2183240/2452/1/1毫克

商品编号： 2452/1

品牌： Tocris Bioscience

市场价： ¥2300.00

美元价： 1380.00

产地：美国(厂家直采)

公司：

产品分类：转运体

公司分类： Transporters

联系Q Q： 3392242852

电话号码： 4000-520-616

电子邮箱： info@ebiomall.com

立即询价

商品介绍

Description:Novel,potentanandamideuptakeinhibitor;inhibitsFAAH

ChemicalName:5-[(1,1'-Biphenyl]-4-yl)methyl]-N,N-dimethyl-1H-tetrazole-1-carboxamide

Purity:≥98%(HPLC)

BIOLOGicalActivityTechnicalDataSolubilityCalculatorsDatasheetsReferences

BiologicalActivity

Novelandhighlypotentblockerofanandamideuptake(IC₅₀=270pM).Inhibitsfattyacidamidehydrolase(FAAH)activity(IC₅₀=12.4nM).Followingi.p.admiNISTrationinrats,increasesbrainanandamideconcentrationandexertsantinociceptiveeffectsinformalinmodelofpain.

LicensingInformation

SoldunderlicensefromEliLillyandCompany

CompoundLibraries

LY2183240isalsoofferedaspartoftheTocriscreenPlus.FindoutmoreaboutcompoundlibrariesavailablefromTocris.

TechnicalData

M.Wt	307.35
Formula	C₁₇H₁₇N₅O
Storage	Storeat+4°C
Purity	≥98%(HPLC)
CASNumber	874902-19-9
PubChemID	11507802
InChIKey	GZNIYOXWFCDBBJ-UHFFFAOYSA-N
Smiles	CN(C)C(=O)N1N=NN=C1CC1=CC=C(C=C1)C1=CC=CC=C1

Thetechnicaldataprovidedaboveisforguidanceonly.ForbatchspecificdatarefertotheCertificateofAnalysis.

AllTocrisproductsareintendedforlaboratoryresearchuseonly.

SolubilityData

	Solvent	MaxConc.mg/mL	MaxConc.mM
Solubility
	DMSO	30.74	100
	ethanol	15.37	50mMwithgentlewarming

PreparingStockSolutions

Thefollowingdataisbasedontheproductmolecularweight307.35.Batchspecificmolecularweightsmayvaryfrombatchtobatchduetosolventofhydration,whichwillaffectthesolventvolumesrequiredtopreparestocksolutions.

Concentration/SolventVolume/Mass	1mg	5mg	10mg
1mM	3.25mL	16.27mL	32.54mL
5mM	0.65mL	3.25mL	6.51mL
10mM	0.33mL	1.63mL	3.25mL
50mM	0.07mL	0.33mL	0.65mL

ProductDatasheets

CertificateofAnalysis/ProductDatasheet

SafetyDatasheet

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