Tocris/Loperamide hydrochloride/0840/1G/1 g-免疫在线蚂蚁淘旗下平台

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商品详细Tocris/Loperamide hydrochloride/0840/1G/1 g

Tocris/Loperamide hydrochloride/0840/1G/1 g

商品编号： 0840/1G

品牌： Tocris Bioscience

市场价： ¥1780.00

美元价： 1068.00

产地：美国(厂家直采)

公司：

产品分类：受体

公司分类： Receptors

联系Q Q： 3392242852

电话号码： 4000-520-616

电子邮箱： info@ebiomall.com

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商品介绍

Description:PeripherallyactingμagoNIST;Ca²⁺channelblocker

ChemicalName:4-(4-Chlorophenyl)-4-hydroxy-N,N-dimethyl-α,α-diphenyl-1-piperidiNEButanamidehydrochloride

Purity:≥99%(HPLC)

BIOLOGicalActivityTechnicalDataSolubilityCalculatorsDatasheetsReferences

BiologicalActivity

Highaffinityμ-opioidreceptoragonistwithperipheralselectivity(K_ivaluesare2,48and1156nMforμ-,δ-andκ-opioidreceptorsrespectively).Antidiarrhoealandantihyperalgesicagent.AlsoaCa²⁺channelblocker;atlowmicromolarconcentrationsitblocksbroadspectrumneuronalHVACa²⁺channelsandathigherconcentrationsitreducesCa²⁺fluxthroughNMDAreceptoroperatedchannels.

TechnicalData

M.Wt	513.51
Formula	C₂₉H₃₃ClN₂O₂.HCl
Storage	StoreatRT
Purity	≥99%(HPLC)
CASNumber	34552-83-5
PubChemID	71420
InChIKey	PGYPOBZJRVSMDS-UHFFFAOYSA-N
Smiles	Cl.CN(C)C(=O)C(CCN1CCC(O)(CC1)C1=CC=C(Cl)C=C1)(C1=CC=CC=C1)C1=CC=CC=C1

Thetechnicaldataprovidedaboveisforguidanceonly.ForbatchspecificdatarefertotheCertificateofAnalysis.

AllTocrisproductsareintendedforlaboratoryresearchuseonly.

SolubilityData

	Solvent	MaxConc.mg/mL	MaxConc.mM
Solubility
	DMSO	10.27	20
	ethanol	10.27	20

PreparingStockSolutions

Thefollowingdataisbasedontheproductmolecularweight513.51.Batchspecificmolecularweightsmayvaryfrombatchtobatchduetosolventofhydration,whichwillaffectthesolventvolumesrequiredtopreparestocksolutions.

Concentration/SolventVolume/Mass	1mg	5mg	10mg
1mM	1.95mL	9.74mL	19.47mL
5mM	0.39mL	1.95mL	3.89mL
10mM	0.19mL	0.97mL	1.95mL
50mM	0.04mL	0.19mL	0.39mL

ProductDatasheets

CertificateofAnalysis/ProductDatasheet

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BiologicalActivity

TechnicalData

SolubilityData

PreparingStockSolutions

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