Biological Activity
High affinity κ agonist with no measured binding at μ or δ sites.
Technical Data
| M. Wt | 358.91 |
| Formula | C21H26N2O.HCl |
| Storage | Store at RT |
| CAS Number | 207452-97-9 |
| PubChem ID | 56972158 |
| InChI Key | BJJKMJWQLJIRGF-VEIFNGETSA-N |
| Smiles | O=C(CC3=CC=CC=C3)N([C@]([C@]2=CC=CC=C2)([H])CN1CCCC1)C.Cl |
The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
All Tocris products are intended for laboratory research use only.
Solubility Data
| Solvent | Max Conc. mg/mL | Max Conc. mM | |
|---|---|---|---|
| Solubility | |||
| DMSO | 8.97 | 25 |
Preparing Stock Solutions
The following data is based on the product molecular weight 358.91. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.
| Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
|---|---|---|---|
| 1 mM | 2.79 mL | 13.93 mL | 27.86 mL |
| 5 mM | 0.56 mL | 2.79 mL | 5.57 mL |
| 10 mM | 0.28 mL | 1.39 mL | 2.79 mL |
| 50 mM | 0.06 mL | 0.28 mL | 0.56 mL |
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Product Datasheets
on-line. Please contact Customer Service
References
References are publications that support the products' biological activity.
Weerawarna et al (1994) Isothiocyanate-substituted κ-selective opioid receptor ligands derived from N-methyl-N-[(1S)-1-phenyl-2-(1-pyrrolidinyl)ethyl]phenylacetamide. J.Med.Chem. 37 2856 PMID: 8071934
Keywords: N-MPPP Hydrochloride, supplier, Selective, κ-opioid, kappa-opioid, agonists, KOP, Receptors, OP2, Kappa, Opioid, Receptors, Kappa, Opioid, Receptors, Tocris Bioscience
