Tocris/MRS 2500 tetraammonium salt/2159/1/1 mg-免疫在线蚂蚁淘旗下平台

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商品详细Tocris/MRS 2500 tetraammonium salt/2159/1/1 mg

Tocris/MRS 2500 tetraammonium salt/2159/1/1 mg

商品编号： 2159/1

品牌： Tocris Bioscience

市场价： ¥6380.00

美元价： 3828.00

产地：美国(厂家直采)

公司：

产品分类：受体

公司分类： Receptors

联系Q Q： 3392242852

电话号码： 4000-520-616

电子邮箱： info@ebiomall.com

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商品介绍

Description:ExtremelypotentandselectiveP2Y₁antagoNIST

ChemicalName:(1R*,2S*)-4-[2-Iodo-6-(methylamino)-9H-purin-9-yl]-2-(phosphonooxy)bicyclo[3.1.0]hexane-1-methanoldihydrogenphosphateestertetraammoniumsalt

Purity:≥96%(HPLC)

BIOLOGicalActivityTechnicalDataSolubilityCalculatorsDatasheetsReferences

BiologicalActivity

HighlypotentandselectiveantagonistoftheplateletP2Y₁receptor(K_i=0.78nM).InhibitsADP-inducedaggregationofhumanplateletswithanIC₅₀valueof0.95nM.InhibitstheupregulationofNTPDase1byATPγS.Preventsthrombusformationinvivo.

LicensingInformation

SoldunderlicensefromtheNIH,USPatent10/169975

TechnicalData

M.Wt	629.29
Formula	C₁₃H₁₈N₅O₈P₂I.4NH₃
Storage	Storeat-20°C
Purity	≥96%(HPLC)
CASNumber	630103-23-0
PubChemID	90488745
InChIKey	FVTFHHDVLNQSME-AVAGOIHISA-N
Smiles	IC4=NC1=C(C(NC)=N4)N=CN1[C@H]2C[C@H](OP(O)(O)=O)[C@@]3(COP(O)(O)=O)[C@@H]2C3.N.N.N.N

Thetechnicaldataprovidedaboveisforguidanceonly.ForbatchspecificdatarefertotheCertificateofAnalysis.

AllTocrisproductsareintendedforlaboratoryresearchuseonly.

SolubilityData

	Solvent	MaxConc.mg/mL	MaxConc.mM
Solubility
Solubility	water	56.12	100

PreparingStockSolutions

Thefollowingdataisbasedontheproductmolecularweight629.29.Batchspecificmolecularweightsmayvaryfrombatchtobatchduetosolventofhydration,whichwillaffectthesolventvolumesrequiredtopreparestocksolutions.

Concentration/SolventVolume/Mass	1mg	5mg	10mg
1mM	1.59mL	7.95mL	15.89mL
5mM	0.32mL	1.59mL	3.18mL
10mM	0.16mL	0.79mL	1.59mL
50mM	0.03mL	0.16mL	0.32mL

ProductDatasheets

CertificateofAnalysis/ProductDatasheet

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BiologicalActivity

LicensingInformation

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SolubilityData

PreparingStockSolutions

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