Biological Activity
Selective P2Y4 receptor agonist (EC50 values are 23, 640, and 740 nM for hP2Y4, hP2Y2 and hP2Y6 respectively).
Technical Data
| M. Wt | 1022.09 |
| Formula | C18H26N3O15P3.4(C2H5)3N |
| Storage | Store at -20°C |
| Purity | ≥99% (HPLC) |
| CAS Number | 1309871-50-8 |
| PubChem ID | 90488925 |
| InChI Key | ZCDZFMKRHPANNI-IHQKQWLFSA-N |
| Smiles | O[C@@H]1[C@@H](COP(OP(OP([O-])([O-])=O)([O-])=O)([O-])=O)O[C@@H](N3C(N/C(C=C3)=NOCCCC2=CC=CC=C2)=O)[C@@H]1O.CC[N+](CC)([H])CC.CC[N+](CC)([H])CC.CC[N+](CC)([H])CC.CC[N+](CC)([H])CC |
The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
All Tocris products are intended for laboratory research use only.
Solubility Data
| Solubility | Soluble in water (supplied pre-dissolved at a concentration of 10mM) |
Preparing Stock Solutions
The following data is based on the product molecular weight 1022.09. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.
| Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
|---|---|---|---|
| 1 mM | 0.98 mL | 4.89 mL | 9.78 mL |
| 5 mM | 0.2 mL | 0.98 mL | 1.96 mL |
| 10 mM | 0.1 mL | 0.49 mL | 0.98 mL |
| 50 mM | 0.02 mL | 0.1 mL | 0.2 mL |
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Product Datasheets
References
References are publications that support the products' biological activity.
Maruoka et al (2011) Pyrimidine nucleotides with 4-alkyloxyimino and terminal tetraphosphate δ-ester modifications as selective agonists of the P2Y4 receptor. J.Med.Chem. 54 4018 PMID: 21528910
Keywords: MRS 4062 triethylammonium salt, supplier, MRS4062, triethylammonium, salt, Selective, P2Y4, agonists, Receptors, Purinergic, purinoceptors, Purinergic, P2Y, Receptors, Purinergic, P2Y, Receptors, Tocris Bioscience
