Tocris/Mps BAY 2a/5562/10/10 mg-免疫在线蚂蚁淘旗下平台

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商品详细Tocris/Mps BAY 2a/5562/10/10 mg

Tocris/Mps BAY 2a/5562/10/10 mg

商品编号： 5562/10

品牌： Tocris Bioscience

市场价： ¥4500.00

美元价： 2700.00

产地：美国(厂家直采)

公司：

产品分类：其它酶

公司分类： Other_enzymes

联系Q Q： 3392242852

电话号码： 4000-520-616

电子邮箱： info@ebiomall.com

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商品介绍

Description:PotentandselectiveMps1kinaseinhibitor

ChemicalName:N-Cyclopropyl-4-[8-[(2-methylpropyl)amino]-6-(5-quinolinyl)imidazo[1,2-a]pyrazin-3-yl]benzamide

Purity:≥98%(HPLC)

BIOLOGicalActivityTechnicalDataSolubilityCalculatorsDatasheetsReferences

BiologicalActivity

PotentandselectiveMps1inhibitor(IC₅₀=1nMforhumanenzyme).SelectiveforMps1overapanelof220kinases.Differentiallyinhibitshumancoloncarcinomacellproliferation.Blockscellcycleprogressionbypreventingspindleassemblycheckpointactivation.Inducesapoptosis.

CompoundLibraries

MpsBAY2aisalsoofferedaspartoftheTocriscreenPlus.FindoutmoreaboutcompoundlibrariesavailablefromTocris.

TechnicalData

M.Wt	476.57
Formula	C₂₉H₂₈N₆O
Storage	Storeat-20°C
Purity	≥98%(HPLC)
CASNumber	1382477-96-4
PubChemID	57381882
InChIKey	MDYKTGNHXNTATG-UHFFFAOYSA-N
Smiles	CC(C)CNC1=NC(C2=CC=CC3=C2C=CC=N3)=CN4C1=NC=C4C5=CC=C(C(NC6CC6)=O)C=C5

Thetechnicaldataprovidedaboveisforguidanceonly.ForbatchspecificdatarefertotheCertificateofAnalysis.

AllTocrisproductsareintendedforlaboratoryresearchuseonly.

SolubilityData

	Solvent	MaxConc.mg/mL	MaxConc.mM
Solubility
	DMSO	47.66	100
	ethanol	47.66	100

PreparingStockSolutions

Thefollowingdataisbasedontheproductmolecularweight476.57.Batchspecificmolecularweightsmayvaryfrombatchtobatchduetosolventofhydration,whichwillaffectthesolventvolumesrequiredtopreparestocksolutions.

Concentration/SolventVolume/Mass	1mg	5mg	10mg
1mM	2.1mL	10.49mL	20.98mL
5mM	0.42mL	2.1mL	4.2mL
10mM	0.21mL	1.05mL	2.1mL
50mM	0.04mL	0.21mL	0.42mL

ProductDatasheets

CertificateofAnalysis/ProductDatasheet

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BiologicalActivity

CompoundLibraries

TechnicalData

SolubilityData

PreparingStockSolutions

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ProductDatasheets