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Tocris Bioscience(优势品牌)
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4000-520-616
当前位置: 首页 > 产品中心 > Receptors > Tocris/NE 100 hydrochloride/3133/10/10 mg
商品详细Tocris/NE 100 hydrochloride/3133/10/10 mg
Tocris/NE 100 hydrochloride/3133/10/10 mg
Tocris/NE 100 hydrochloride/3133/10/10 mg
商品编号: 3133/10
品牌: Tocris Bioscience
市场价: ¥3100.00
美元价: 1860.00
产地: 美国(厂家直采)
公司:
产品分类: 受体
公司分类: Receptors
联系Q Q: 3392242852
电话号码: 4000-520-616
电子邮箱: info@ebiomall.com
商品介绍
Description:Selectiveσ1antagoNIST
ChemicalName:4-Methoxy-3-(2-phenylethoxy)-N,N-dipropylbenzeneethanaminehydrochloride
Purity:≥98%(HPLC)
BIOLOGicalActivityTechnicalDataSolubilityCalculatorsDatasheetsReferences

BiologicalActivity

Potentandselectiveσ1receptorantagonist(Ki=0.86nM)thatdisplays>55-foldselectivityoverσ2receptorsand>6000-foldselectivityoverD1,D2,5-HT1A,5-HT2andPCPreceptors.ExhibitsreversIBLebinding(Kd=1.2nM)anddisplaysantipsychoticactivityinvivo.Orallyactive.

CompoundLibraries

NE100hydrochlorideisalsoofferedaspartoftheTocriscreenPlus.FindoutmoreaboutcompoundlibrariesavailablefromTocris.

TechnicalData

M.Wt391.97
FormulaC23H33NO2.HCl
StorageStoreat-20°C
Purity≥98%(HPLC)
CASNumber149409-57-4
PubChemID9952420
InChIKeyZHGMDXSHODHWHV-UHFFFAOYSA-N
SmilesCCCN(CCC)CCC1=CC=C(OC)C(OCCC2=CC=CC=C2)=C1.Cl

Thetechnicaldataprovidedaboveisforguidanceonly.ForbatchspecificdatarefertotheCertificateofAnalysis.

AllTocrisproductsareintendedforlaboratoryresearchuseonly.

SolubilityData

SolventMaxConc.mg/mLMaxConc.mM
Solubility
DMSO39.2100
water9.825

PreparingStockSolutions

Thefollowingdataisbasedontheproductmolecularweight391.97.Batchspecificmolecularweightsmayvaryfrombatchtobatchduetosolventofhydration,whichwillaffectthesolventvolumesrequiredtopreparestocksolutions.

Concentration/SolventVolume/Mass1mg5mg10mg
1mM2.55mL12.76mL25.51mL
5mM0.51mL2.55mL5.1mL
10mM0.26mL1.28mL2.55mL
50mM0.05mL0.26mL0.51mL

ProductDatasheets

CertificateofAnalysis/ProductDatasheet
SafetyDatasheet