Tocris/PD 135158/2608/50/50 mg-免疫在线蚂蚁淘旗下平台

当前位置：首页 > 产品中心 > Receptors > Tocris/PD 135158/2608/50/50 mg

商品详细Tocris/PD 135158/2608/50/50 mg

Tocris/PD 135158/2608/50/50 mg

商品编号： 2608/50

品牌： Tocris Bioscience

市场价： ¥20900.00

美元价： 12540.00

产地：美国(厂家直采)

公司：

产品分类：受体

公司分类： Receptors

联系Q Q： 3392242852

电话号码： 4000-520-616

电子邮箱： info@ebiomall.com

立即询价

商品介绍

Description:PotentandselectiveCCK₂antagoNIST

AlternativeNames:CAM1028

ChemicalName:4-[[(1R)-2-[[(2R)-3-(1H-Indol-3-yl)-2-methyl-1-oxo-2-[[[[(1S,2R,4S)-1,7,7-trimethylbicyclo[2.2.1]hept-2-yl]oxy]carbonyl]amino]propyl]amino]-1-phenylethyl]amino]-4-oxobutanoicacid

Purity:≥98%(HPLC)

BIOLOGicalActivityTechnicalDataSolubilityCalculatorsDatasheetsReferences

BiologicalActivity

Potentandselective,nonpeptideCCK₂receptorantagonist(IC₅₀valuesare2.8and1232nMforCCK₂andCCK₁respectively)thatdisplaysnegligIBLeaffinityatGABA_A,benzodiazepine,substanceP,neurotensin,opioid,bradykininand5-HT₃receptors(IC₅₀>10μM).Exhibitsanxiolyticactivityinelevatedplusmazeandsocialinteractiontestsandincreasesfoodintakeinrats.

TechnicalData

M.Wt	616.76
Formula	C₃₅H₄₄N₄O₆
Storage	Storeat+4°C
Purity	≥98%(HPLC)
CASNumber	130285-87-9
PubChemID	44385784
InChIKey	NNTPEWZUKRSTMM-CFHPNWNBSA-N
Smiles	C[C@](NC(OC3C4(C)CCC(C(C)4C)C3)=O)(C(NC[C@@H]([C@]5=CC=CC=C5)NC(CCC(O)=O)=O)=O)CC2=CNC1=CC=CC=C12

Thetechnicaldataprovidedaboveisforguidanceonly.ForbatchspecificdatarefertotheCertificateofAnalysis.

AllTocrisproductsareintendedforlaboratoryresearchuseonly.

SolubilityData

	Solvent	MaxConc.mg/mL	MaxConc.mM
Solubility
Solubility	DMSO	61.68	100

PreparingStockSolutions

Thefollowingdataisbasedontheproductmolecularweight616.76.Batchspecificmolecularweightsmayvaryfrombatchtobatchduetosolventofhydration,whichwillaffectthesolventvolumesrequiredtopreparestocksolutions.

Concentration/SolventVolume/Mass	1mg	5mg	10mg
1mM	1.62mL	8.11mL	16.21mL
5mM	0.32mL	1.62mL	3.24mL
10mM	0.16mL	0.81mL	1.62mL
50mM	0.03mL	0.16mL	0.32mL

ProductDatasheets

CertificateofAnalysis/ProductDatasheet

SafetyDatasheet

Selectanotherlanguage:

BiologicalActivity

TechnicalData

SolubilityData

PreparingStockSolutions

MolarityCalculator

ReconstitutionCalculator

DilutionCalculator

ProductDatasheets