Biological Activity
A potent analgesic and nootropic agent. Increases release of acetylcholine.
Technical Data
| M. Wt | 468.34 |
| Formula | C17H22BrNO2.C4H4O4 |
| Storage | Store at RT |
| CAS Number | 155649-00-6 |
| PubChem ID | 46905315 |
| InChI Key | VBUSCULTLLOSLM-BTJKTKAUSA-N |
| Smiles | OC(=O)C=C/C(O)=O.CC(C(=O)OC1CC2CCC(C1)N2C)C1=CC=C(Br)C=C1 |
The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
All Tocris products are intended for laboratory research use only.
Solubility Data
| Solvent | Max Conc. mg/mL | Max Conc. mM | |
|---|---|---|---|
| Solubility | |||
| DMSO | 46.83 | 100 |
Preparing Stock Solutions
The following data is based on the product molecular weight 468.34. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.
| Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
|---|---|---|---|
| 1 mM | 2.14 mL | 10.68 mL | 21.35 mL |
| 5 mM | 0.43 mL | 2.14 mL | 4.27 mL |
| 10 mM | 0.21 mL | 1.07 mL | 2.14 mL |
| 50 mM | 0.04 mL | 0.21 mL | 0.43 mL |
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Product Datasheets
References
References are publications that support the products' biological activity.
Ghelardini et al (1998) Antinociceptive and antiamnesic properties of the presynaptic cholinergic amplifier PG-9. J.Pharmacol.Exp.Ther. 284 806 PMID: 9495837
Gualtieri et al (1994) Presynaptic cholinergic modulators as potent cognition enhancers and analgesic drugs. 1. Tropic and 2-phenylpropionic acid esters. J.Med.Chem. 37 1704 PMID: 8201605
Keywords: PG-9 maleate, supplier, Presynaptic, cholinergic, modulators, Acetylcholine, Nicotinic, Receptors, nAChR, Muscarinic, release, Other, Acetylcholine, Non-selective, Muscarinics, Other, Acetylcholine, Tocris Bioscience
