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Tocris Bioscience(优势品牌)
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当前位置: 首页 > 产品中心 > Receptors > Tocris/R-96544 hydrochloride/1742/10/10 mg
商品详细Tocris/R-96544 hydrochloride/1742/10/10 mg
Tocris/R-96544 hydrochloride/1742/10/10 mg
Tocris/R-96544 hydrochloride/1742/10/10 mg
商品编号: 1742/10
品牌: Tocris Bioscience
市场价: ¥3380.00
美元价: 2028.00
产地: 美国(厂家直采)
公司:
产品分类: 受体
公司分类: Receptors
联系Q Q: 3392242852
电话号码: 4000-520-616
电子邮箱: info@ebiomall.com
商品介绍
Description:Potent,selective5-HT2AantagoNIST
ChemicalName:(2R,4R)-5-[2-[2-[2-(3-Methoxyphenyl)ethyl]phenoxy]ethyl]-1-methyl-3-pyrrolidinolhydrochloride
Purity:≥99%(HPLC)
BIOLOGicalActivityTechnicalDataSolubilityCalculatorsDatasheetsReferences

BiologicalActivity

Potent,selective5-HT2receptorantagonist;displayssomeselectivityfor5-HT2Areceptors(Ki=1.6nM).IC50valuesare2.2,310,2400,3700,>5000and>5000nMfor5-HT2,α1-adrenergic,D2dopamine,5-HT1,5-HT3andβ-adrenergicreceptorsrespectively.Inhibits5-HT-inducedplateletaggregationandpressorresponsesinvivo.

CompoundLibraries

R-96544hydrochlorideisalsoofferedaspartoftheTocriscreenPlus.FindoutmoreaboutcompoundlibrariesavailablefromTocris.

TechnicalData

M.Wt391.94
FormulaC22H29NO3.HCl
StorageStoreatRT
Purity≥99%(HPLC)
CASNumber167144-80-1
PubChemID10668210
InChIKeyOUKRSTJUAQEATQ-GZJHNZOKSA-N
SmilesCl[H].COC1=CC=CC(CCC2=C(OCC[C@@H]3C[C@@H](O)CN3C)C=CC=C2)=C1

Thetechnicaldataprovidedaboveisforguidanceonly.ForbatchspecificdatarefertotheCertificateofAnalysis.

AllTocrisproductsareintendedforlaboratoryresearchuseonly.

SolubilityData

SolventMaxConc.mg/mLMaxConc.mM
Solubility
DMSO39.19100
water39.19100

PreparingStockSolutions

Thefollowingdataisbasedontheproductmolecularweight391.94.Batchspecificmolecularweightsmayvaryfrombatchtobatchduetosolventofhydration,whichwillaffectthesolventvolumesrequiredtopreparestocksolutions.

Concentration/SolventVolume/Mass1mg5mg10mg
1mM2.55mL12.76mL25.51mL
5mM0.51mL2.55mL5.1mL
10mM0.26mL1.28mL2.55mL
50mM0.05mL0.26mL0.51mL

ProductDatasheets

CertificateofAnalysis/ProductDatasheet
SafetyDatasheet