Tocris/TC Mps1 12/4750/10/10 mg-免疫在线蚂蚁淘旗下平台

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商品详细Tocris/TC Mps1 12/4750/10/10 mg

Tocris/TC Mps1 12/4750/10/10 mg

商品编号： 4750/10

品牌： Tocris Bioscience

市场价： ¥3980.00

美元价： 2388.00

产地：美国(厂家直采)

公司：

产品分类：其它酶

公司分类： Other_enzymes

联系Q Q： 3392242852

电话号码： 4000-520-616

电子邮箱： info@ebiomall.com

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商品介绍

Description:PotentandselectiveMps1kinaseinhibitor

ChemicalName:4-[[4-Amino-5-cyano-6-[(1,1-dimethylethyl)amino]-2-pyridinyl]amino]benzamide

Purity:≥99%(HPLC)

BIOLOGicalActivityTechnicalDataSolubilityCalculatorsDatasheetsReferences

BiologicalActivity

Potentandselectivemonopolarspindle1(Mps1)inhibitor(IC₅₀=6.4nM).SelectiveforMps1overapanelof95kinasesincludingJNK.InhibitsA549lungcarcinomacellproliferationandattenuatesA549cellxenograftgrowthinmice.Orallyactive.

CompoundLibraries

TCMps112isalsoofferedaspartoftheTocriscreenPlusandTocriscreenKinaseInhibitorToolboxII.FindoutmoreaboutcompoundlibrariesavailablefromTocris.

TechnicalData

M.Wt	324.38
Formula	C₁₇H₂₀N₆O
Storage	Storeat+4°C
Purity	≥99%(HPLC)
CASNumber	1206170-62-8
PubChemID	70682875
InChIKey	XDEFNAWAKYQBQY-UHFFFAOYSA-N
Smiles	NC1=C(C#N)C(NC(C)(C)C)=NC(NC2=CC=C(C(N)=O)C=C2)=C1

Thetechnicaldataprovidedaboveisforguidanceonly.ForbatchspecificdatarefertotheCertificateofAnalysis.

AllTocrisproductsareintendedforlaboratoryresearchuseonly.

SolubilityData

	Solvent	MaxConc.mg/mL	MaxConc.mM
Solubility
	DMSO	32.44	100
	ethanol	6.49	20mMwithgentlewarming

PreparingStockSolutions

Thefollowingdataisbasedontheproductmolecularweight324.38.Batchspecificmolecularweightsmayvaryfrombatchtobatchduetosolventofhydration,whichwillaffectthesolventvolumesrequiredtopreparestocksolutions.

Concentration/SolventVolume/Mass	1mg	5mg	10mg
1mM	3.08mL	15.41mL	30.83mL
5mM	0.62mL	3.08mL	6.17mL
10mM	0.31mL	1.54mL	3.08mL
50mM	0.06mL	0.31mL	0.62mL

ProductDatasheets

CertificateofAnalysis/ProductDatasheet

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BiologicalActivity

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