Tocris/TCS 1102/3818/10/10毫克-免疫在线蚂蚁淘旗下平台

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Tocris/TCS 1102/3818/10/10毫克

商品编号： 3818/10

品牌： Tocris Bioscience

市场价： ¥3180.00

美元价： 1908.00

产地：美国(厂家直采)

公司：

产品分类：受体

公司分类： Receptors

联系Q Q： 3392242852

电话号码： 4000-520-616

电子邮箱： info@ebiomall.com

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商品介绍

Description:Potent,dualorexinreceptorantagoNIST

ChemicalName:N-[1,1'-Biphenyl]-2-yl-1-[2-[(1-methyl-1H-benzimidazol-2-yl)thio]acetyl-2-pyrrolidinedicarboxamide

Purity:≥98%(HPLC)

BIOLOGicalActivityTechnicalDataSolubilityCalculatorsDatasheetsReferences

BiologicalActivity

Potent,dualorexinreceptorantagonist(K_ivaluesare0.2and3nMforOX₂andOX₁receptorsrespectively).InhibitsADL-orexinB-mediatedlocomotionfollowingi.p.administrationinvivoandblocksorexin-A(Cat.No.1455)mediatedincreasesinfeedingbehaviour.Brainpenetrant.

LicensingInformation

ManufacturedandsoldunderlicensefromMerck&Co.,Inc.forusesolelyforpreclinicalresearchpurposes(ie:notforadministrationtoorotheruseinhumans)

TechnicalData

M.Wt	470.59
Formula	C₂₇H₂₆N₄O₂S
Storage	StoreatRT
Purity	≥98%(HPLC)
CASNumber	916141-36-1
PubChemID	11960895
InChIKey	YSBGRVXJEMSEQY-DEOSSOPVSA-N
Smiles	O=C(CSC2=NC(C=CC=C5)=C5N2C)N1CCC[C@H]1[C@](NC3=CC=CC=C3C4=CC=CC=C4)=O

Thetechnicaldataprovidedaboveisforguidanceonly.ForbatchspecificdatarefertotheCertificateofAnalysis.

AllTocrisproductsareintendedforlaboratoryresearchuseonly.

SolubilityData

	Solvent	MaxConc.mg/mL	MaxConc.mM
Solubility
	DMSO	47.06	100
	ethanol	47.06	100

PreparingStockSolutions

Thefollowingdataisbasedontheproductmolecularweight470.59.Batchspecificmolecularweightsmayvaryfrombatchtobatchduetosolventofhydration,whichwillaffectthesolventvolumesrequiredtopreparestocksolutions.

Concentration/SolventVolume/Mass	1mg	5mg	10mg
1mM	2.12mL	10.62mL	21.25mL
5mM	0.42mL	2.12mL	4.25mL
10mM	0.21mL	1.06mL	2.12mL
50mM	0.04mL	0.21mL	0.42mL

ProductDatasheets

CertificateofAnalysis/ProductDatasheet

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BiologicalActivity

LicensingInformation

TechnicalData

SolubilityData

PreparingStockSolutions

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