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商品详细Tocris/Tiplaxtinin/5565/10/10 mg

Tocris/Tiplaxtinin/5565/10/10 mg

商品编号： 5565/10

品牌： Tocris Bioscience

市场价： ¥2380.00

美元价： 1428.00

产地：美国(厂家直采)

公司：

产品分类：蛋白酶类

公司分类： protease

联系Q Q： 3392242852

电话号码： 4000-520-616

电子邮箱： info@ebiomall.com

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商品介绍

Description:Plasminogenactivatorinhibitor-1(PAI-1)inhibitor

AlternativeNames:PAI039,tiplasinin

ChemicalName:α-Oxo-1-(phenylmethyl)-5-[4-(trifluoromethoxy)phenyl]-1H-indole-3-aceticacid

Purity:≥98%(HPLC)

BIOLOGicalActivityTechnicalDataSolubilityCalculatorsDatasheetsReferences

BiologicalActivity

Plasminogenactivatorinhibitor-1(PAI-1)inhibitor(IC₅₀=2.7μM).Inducesvascularsmoothmusclecellapoptosisinvitroandreducescarotidarteryneointimalformationinaratvascularinjurymodel.Promotesthrombolysisinratanddogmodelsofacutearterialthrombosis.Orallyavailable.

CompoundLibraries

TiplaxtininisalsoofferedaspartoftheTocriscreenPlus.FindoutmoreaboutcompoundlibrariesavailablefromTocris.

TechnicalData

M.Wt	439.38
Formula	C₂₄H₁₆F₃NO₄
Storage	Storeat+4°C
Purity	≥98%(HPLC)
CASNumber	393105-53-8
PubChemID	6450819
InChIKey	ODXQFEWQSHNQNI-UHFFFAOYSA-N
Smiles	O=C(C(O)=O)C2=CN(CC3=CC=CC=C3)C1=CC=C(C4=CC=C(OC(F)(F)F)C=C4)C=C12

Thetechnicaldataprovidedaboveisforguidanceonly.ForbatchspecificdatarefertotheCertificateofAnalysis.

AllTocrisproductsareintendedforlaboratoryresearchuseonly.

SolubilityData

	Solvent	MaxConc.mg/mL	MaxConc.mM
Solubility
	DMSO	43.94	100
	ethanol	43.94	100

PreparingStockSolutions

Thefollowingdataisbasedontheproductmolecularweight439.38.Batchspecificmolecularweightsmayvaryfrombatchtobatchduetosolventofhydration,whichwillaffectthesolventvolumesrequiredtopreparestocksolutions.

Concentration/SolventVolume/Mass	1mg	5mg	10mg
1mM	2.28mL	11.38mL	22.76mL
5mM	0.46mL	2.28mL	4.55mL
10mM	0.23mL	1.14mL	2.28mL
50mM	0.05mL	0.23mL	0.46mL

ProductDatasheets

CertificateofAnalysis/ProductDatasheet

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BiologicalActivity

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TechnicalData

SolubilityData

PreparingStockSolutions

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