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当前位置: 首页 > 产品中心 > Receptors > Tocris/Trap 101/2508/10/10 mg
商品详细Tocris/Trap 101/2508/10/10 mg
Tocris/Trap 101/2508/10/10 mg
Tocris/Trap 101/2508/10/10 mg
商品编号: 2508/10
品牌: Tocris Bioscience
市场价: ¥3780.00
美元价: 2268.00
产地: 美国(厂家直采)
公司:
产品分类: 受体
公司分类: Receptors
联系Q Q: 3392242852
电话号码: 4000-520-616
电子邮箱: info@ebiomall.com
商品介绍
Description:PotentandselectiveNOPantagoNIST;activeinvivo
ChemicalName:1-[1-(Cyclooctylmethyl)-1,2,3,6-tetrahydro-5-(hydroxymethyl)-4-pyridinyl]-3-ethyl-1,3-dihydro-2H-benzimidazol-2-onehydrochloride
Purity:≥98%(HPLC)
BIOLOGicalActivityTechnicalDataSolubilityCalculatorsDatasheetsReferences

BiologicalActivity

Potentandselectivenociceptin/orphaninFQ(NOP)receptorantagonist(pA2=7.75).DisplaysselectivityforNOPreceptorsoverclassicalopioidreceptors(pKivaluesare8.65,6.60,6.14and<5forNOP,μ-,κ-,andδ-opioidreceptorsrespectively).AttenuatesmotordeficitsinaratmodelofParkinson'sDisease.Activeinvivo.

CompoundLibraries

Trap101isalsoofferedaspartoftheTocriscreenPlus.FindoutmoreaboutcompoundlibrariesavailablefromTocris.

TechnicalData

M.Wt434.02
FormulaC24H35N3O2.HCl
StorageStoreat+4°C
Purity≥98%(HPLC)
CASNumber1216621-00-9
PubChemID56972178
InChIKeyYEVMLMQAMCKVSC-UHFFFAOYSA-N
SmilesCl.CCN1C(=O)N(C2=CC=CC=C12)C1=C(CO)CN(CC2CCCCCCC2)CC1

Thetechnicaldataprovidedaboveisforguidanceonly.ForbatchspecificdatarefertotheCertificateofAnalysis.

AllTocrisproductsareintendedforlaboratoryresearchuseonly.

SolubilityData

SolventMaxConc.mg/mLMaxConc.mM
Solubility
DMSO21.750

PreparingStockSolutions

Thefollowingdataisbasedontheproductmolecularweight434.02.Batchspecificmolecularweightsmayvaryfrombatchtobatchduetosolventofhydration,whichwillaffectthesolventvolumesrequiredtopreparestocksolutions.

Concentration/SolventVolume/Mass1mg5mg10mg
1mM2.3mL11.52mL23.04mL
5mM0.46mL2.3mL4.61mL
10mM0.23mL1.15mL2.3mL
50mM0.05mL0.23mL0.46mL

ProductDatasheets

CertificateofAnalysis/ProductDatasheet
SafetyDatasheet