Tocris/XCT 790/3928/10/10毫克-免疫在线蚂蚁淘旗下平台

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Tocris/XCT 790/3928/10/10毫克

商品编号： 3928/10

品牌： Tocris Bioscience

市场价： ¥3380.00

美元价： 2028.00

产地：美国(厂家直采)

公司：

产品分类：受体

公司分类： Receptors

联系Q Q： 3392242852

电话号码： 4000-520-616

电子邮箱： info@ebiomall.com

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商品介绍

Description:SelectiveERRαantagoNIST/inverseagonist

ChemicalName:3-[4-(2,4-Bis-trifluoromethylbenzyloxy)-3-methoxyphenyl]-2-cyano-N-(5-trifluoromethyl-1,3,4-thiADIazol-2-yl)acrylamide

Purity:≥99%(HPLC)

BIOLOGicalActivityTechnicalDataSolubilityCalculatorsDatasheetsReferences

BiologicalActivity

SelectiveERRαantagonist/inverseagonist(IC₅₀=~400nM).DisplaysnoantagonistactivityatERRγorERαatconcentrationsbelow10μM.InterfereswithPPARγcoactivator-1α(PGC-1α)/ERRα-dependentsignaling:inhibitsPGC-1αinductionofERRαandMAO-BgeneexpressionanddownregulatestheconstitutivetranscriptionalactivityofERRαinnumerouscelllines.

TechnicalData

M.Wt	596.42
Formula	C₂₃H₁₃F₉N₄O₃S
Storage	Storeat+4°C
Purity	≥99%(HPLC)
CASNumber	725247-18-7
PubChemID	6918788
InChIKey	HQFNFOOGGLSBBT-AWNIVKPZSA-N
Smiles	O=C(NC3=NN=C(C(F)(F)F)S3)/C(C#N)=C/C(C=C2OC)=CC=C2OCC1=C(C(F)(F)F)C=C(C(F)(F)F)C=C1

Thetechnicaldataprovidedaboveisforguidanceonly.ForbatchspecificdatarefertotheCertificateofAnalysis.

AllTocrisproductsareintendedforlaboratoryresearchuseonly.

SolubilityData

	Solvent	MaxConc.mg/mL	MaxConc.mM
Solubility
Solubility	DMSO	5.96	10mMwithgentlewarming

PreparingStockSolutions

Thefollowingdataisbasedontheproductmolecularweight596.42.Batchspecificmolecularweightsmayvaryfrombatchtobatchduetosolventofhydration,whichwillaffectthesolventvolumesrequiredtopreparestocksolutions.

Concentration/SolventVolume/Mass	1mg	5mg	10mg
1mM	1.68mL	8.38mL	16.77mL
5mM	0.34mL	1.68mL	3.35mL
10mM	0.17mL	0.84mL	1.68mL
50mM	0.03mL	0.17mL	0.34mL

ProductDatasheets

CertificateofAnalysis/ProductDatasheet

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BiologicalActivity

TechnicalData

SolubilityData

PreparingStockSolutions

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