Tocris/AZ PFKFB3 26/5675/50/50 mg-免疫在线蚂蚁淘旗下平台

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商品详细Tocris/AZ PFKFB3 26/5675/50/50 mg

Tocris/AZ PFKFB3 26/5675/50/50 mg

商品编号： 5675/50

品牌： Tocris Bioscience

市场价： ¥10900.00

美元价： 6540.00

产地：美国(厂家直采)

公司：

产品分类：其它酶

公司分类： Other_enzymes

联系Q Q： 3392242852

电话号码： 4000-520-616

电子邮箱： info@ebiomall.com

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商品介绍

Description:PotentandselectivePFKFB3inhibitor

ChemicalName:(2S)-N-[4-[[3-Cyano-1-(2-methylpropyl)-1H-indol-5-yl]oxy]phenyl]-2-pyrrolidinecarboxamide

Purity:≥98%(HPLC)

BIOLOGicalActivityTechnicalDataSolubilityCalculatorsDatasheetsReferences

BiologicalActivity

PotentandselectivePFKFB3inhibitor(IC₅₀=0.023μM).SelectiveforPFKFB3overPFKFB2andPFKFB1isoforms(IC₅₀valuesare0.382μMand2.06μM,respectively).Reduceslevelsoffructose-1,6-bisphosphateinA549cells(IC₅₀=0.343μM).Exhibitsnosignificantinhibitionofotherkinases.

TechnicalData

M.Wt	402.49
Formula	C₂₄H₂₆N₄O₂
Storage	Storeat-20°C
Purity	≥98%(HPLC)
CASNumber	1704740-52-2
PubChemID	118735769
InChIKey	OOGHGWKBJXQNEJ-QFIPXVFZSA-N
Smiles	N#CC1=CN(CC(C)C)C2=C1C=C(OC3=CC=C(NC([C@H]4NCCC4)=O)C=C3)C=C2

Thetechnicaldataprovidedaboveisforguidanceonly.ForbatchspecificdatarefertotheCertificateofAnalysis.

AllTocrisproductsareintendedforlaboratoryresearchuseonly.

SolubilityData

	Solvent	MaxConc.mg/mL	MaxConc.mM
Solubility
	DMSO	40.25	100
	ethanol	40.25	100

PreparingStockSolutions

Thefollowingdataisbasedontheproductmolecularweight402.49.Batchspecificmolecularweightsmayvaryfrombatchtobatchduetosolventofhydration,whichwillaffectthesolventvolumesrequiredtopreparestocksolutions.

Concentration/SolventVolume/Mass	1mg	5mg	10mg
1mM	2.48mL	12.42mL	24.85mL
5mM	0.5mL	2.48mL	4.97mL
10mM	0.25mL	1.24mL	2.48mL
50mM	0.05mL	0.25mL	0.5mL

ProductDatasheets

CertificateofAnalysis/ProductDatasheet

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BiologicalActivity

TechnicalData

SolubilityData

PreparingStockSolutions

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