Tocris/A 922500/3587/10/10 mg-免疫在线蚂蚁淘旗下平台

当前位置：首页 > 产品中心 > Other_enzymes > Tocris/A 922500/3587/10/10 mg

商品详细Tocris/A 922500/3587/10/10 mg

Tocris/A 922500/3587/10/10 mg

商品编号： 3587/10

品牌： Tocris Bioscience

市场价： ¥6180.00

美元价： 3708.00

产地：美国(厂家直采)

公司：

产品分类：其它酶

公司分类： Other_enzymes

联系Q Q： 3392242852

电话号码： 4000-520-616

电子邮箱： info@ebiomall.com

立即询价

商品介绍

Description:PotentDGAT-1inhibitor

AlternativeNames:DGAT-1Inhibitor4a

ChemicalName:(1R,2R)-2-[[4'-[[Phenylamino)carbonyl]amino][1,1'-biphenyl]-4-yl]carbonyl]cyclopentanecarboxylicacid

Purity:≥98%(HPLC)

BIOLOGicalActivityTechnicalDataSolubilityCalculatorsDatasheetsReferences

BiologicalActivity

Diacylglycerolacyltransferase1(DGAT-1)inhibitor(IC₅₀valuesare7and24nMathumanandmouseDGAT-1respectively)thatisdevoidofactivityatDGAT-2,ACAT1orACAT2.Inducessignificantweightlosswithoutalteringfoodintake,anddecreasesliverandplasmatriglyceridelevelsinvivo.Orallyactive.

CompoundLibraries

A922500isalsoofferedaspartoftheTocriscreenPlus.FindoutmoreaboutcompoundlibrariesavailablefromTocris.

TechnicalData

M.Wt	428.48
Formula	C₂₆H₂₄N₂O₄
Storage	Desiccateat+4°C
Purity	≥98%(HPLC)
CASNumber	959122-11-3
PubChemID	24768261
InChIKey	BOZRFEQDOFSZBV-DHIUTWEWSA-N
Smiles	O=[C@]([C@@H]3CCC[C@H]3[C@@](O)=O)C(C=C2)=CC=C2C1=CC=C(NC(NC4=CC=CC=C4)=O)C=C1

Thetechnicaldataprovidedaboveisforguidanceonly.ForbatchspecificdatarefertotheCertificateofAnalysis.

AllTocrisproductsareintendedforlaboratoryresearchuseonly.

SolubilityData

	Solvent	MaxConc.mg/mL	MaxConc.mM
Solubility
Solubility	DMSO	21.42	50

PreparingStockSolutions

Thefollowingdataisbasedontheproductmolecularweight428.48.Batchspecificmolecularweightsmayvaryfrombatchtobatchduetosolventofhydration,whichwillaffectthesolventvolumesrequiredtopreparestocksolutions.

Concentration/SolventVolume/Mass	1mg	5mg	10mg
1mM	2.33mL	11.67mL	23.34mL
5mM	0.47mL	2.33mL	4.67mL
10mM	0.23mL	1.17mL	2.33mL
50mM	0.05mL	0.23mL	0.47mL

ProductDatasheets

CertificateofAnalysis/ProductDatasheet

SafetyDatasheet

Selectanotherlanguage:

BiologicalActivity

CompoundLibraries

TechnicalData

SolubilityData

PreparingStockSolutions

MolarityCalculator

ReconstitutionCalculator

DilutionCalculator

ProductDatasheets