Tocris/A 987306/3640/10/10毫克-免疫在线蚂蚁淘旗下平台

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商品详细Tocris/A 987306/3640/10/10毫克

Tocris/A 987306/3640/10/10毫克

商品编号： 3640/10

品牌： Tocris Bioscience

市场价： ¥4700.00

美元价： 2820.00

产地：美国(厂家直采)

公司：

产品分类：受体

公司分类： Receptors

联系Q Q： 3392242852

电话号码： 4000-520-616

电子邮箱： info@ebiomall.com

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商品介绍

Description:PotentandselectiveH₄receptorantagoNIST

ChemicalName:(±)-(7aR*,11aR*)-5,6,7a,8,9,10,11,11a-Octahydro-4-(1-piperazinyl)-benzofuran[2,3-h]quinazolin-2-amine

Purity:≥98%(HPLC)

BIOLOGicalActivityTechnicalDataSolubilityCalculatorsDatasheetsReferences

BiologicalActivity

PotenthistamineH₄receptorantagonist(pK_ivaluesare8.24and8.47inhumanandratH₄receptorsrespectively).Displays162-fold,620-fold,and>1600-foldselectivityoverhumanH₃,H₁andH₂receptors.Blockszymosan-inducedneutrophilrefluxandattenuatesthermalhypersensitivityinvivo(ED₅₀=42μmol/kg,ip).

CompoundLibraries

A987306isalsoofferedaspartoftheTocriscreenPlus.FindoutmoreaboutcompoundlibrariesavailablefromTocris.

TechnicalData

M.Wt	327.42
Formula	C₁₈H₂₅N₅O
Storage	Storeat-20°C
Purity	≥98%(HPLC)
CASNumber	1082954-71-9
PubChemID	25109291
InChIKey	DJKJVWJQAVGLHJ-YPMHNXCESA-N
Smiles	NC3=NC1=C(C(N4CCNCC4)=N3)CCC2=C1[C@@](CCCC5)([H])[C@@]5([H])O2

Thetechnicaldataprovidedaboveisforguidanceonly.ForbatchspecificdatarefertotheCertificateofAnalysis.

AllTocrisproductsareintendedforlaboratoryresearchuseonly.

SolubilityData

	Solvent	MaxConc.mg/mL	MaxConc.mM
Solubility
	DMSO	32.74	100
	ethanol	32.74	100

PreparingStockSolutions

Thefollowingdataisbasedontheproductmolecularweight327.42.Batchspecificmolecularweightsmayvaryfrombatchtobatchduetosolventofhydration,whichwillaffectthesolventvolumesrequiredtopreparestocksolutions.

Concentration/SolventVolume/Mass	1mg	5mg	10mg
1mM	3.05mL	15.27mL	30.54mL
5mM	0.61mL	3.05mL	6.11mL
10mM	0.31mL	1.53mL	3.05mL
50mM	0.06mL	0.31mL	0.61mL

ProductDatasheets

CertificateofAnalysis/ProductDatasheet

SafetyDatasheet

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BiologicalActivity

CompoundLibraries

TechnicalData

SolubilityData

PreparingStockSolutions

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